prof. dr hab. Andrzej Bojarski

prof. dr hab. Andrzej Bojarski

+48 12 6623365
pokój 325
Zakład Chemii Leków

Dokonania naukowe

  • Publikacje

Synthesis and biological evaluation of new multi-target 3-(1<i>H</i>-indol-3-yl)pyrrolidine-2,5-dione derivatives with potential antidepressant effect

Autorzy: Wrobel, Martyna Z., Chodkowski, Andrzej, Herold, Franciszek, Marciniak, Monika, Dawidowski, Maciej, Siwek, Agata, Starowicz, Gabriela, Stachowicz, Katarzyna, Szewczyk, Bernadeta, Nowak, Gabriel, Belka, Mariusz, Baczek, Tomasz, Satala, Grzegorz, Bojarski, Andrzej J., Turlo, Jadwiga

DOI: 10.1016/J.EJMECH.2019.111736
Date: 2019-01-01

Oncotoxic Properties of Serotonin Transporter Inhibitors and 5-HT<sub>1A</sub> Receptor Ligands

Autorzy: Jarosław Walory, Lidia Mielczarek, Małgorzata Jarończyk, Mirosława Koronkiewicz, Jerzy Kossakowski, Ryszard Bugno, Andrzej Bojarski, Zdzisław Chilmonczyk

DOI: 10.3390/ijms19103260
Date: 2018-10-01

Substructural Connectivity Fingerprint and Extreme Entropy Machines—A New Method of Compound Representation and Analysis

Autorzy:

DOI: 10.3390/molecules23061242
Date: 2018-05-01

Fingerprint-Based Machine Learning Approach to Identify Potent and Selective 5-HT<sub>2B</sub>R Ligands

Autorzy:

DOI: 10.3390/molecules23051137
Date: 2018-05-01

Search for a 5-CT alternative. In vitro and in vivo evaluation of novel pharmacological tools: 3-(1-alkyl-1H-imidazol-5-yl)-1H-indole-5-carboxamides, low-basicity 5-HT7 receptor agonists

Autorzy: Latacz, Gniewomir, Hogendorf, Adam S., Hogendorf, Agata, Lubelska, Annamaria, Wieronska, Joanna M., Wozniak, Monika, Cieslik, Paulina, Kiec-Kononowicz, Katarzyna, Handzlik, Jadwiga, Bojarski, Andrzej J.

DOI: 10.1039/C8MD00313K
Date: 2018-01-01

Selective inhibition of human cathepsin S by 2,4,6-trisubstituted 1,3,5-triazine analogs

Autorzy: Tber, Z., Wartenberg, M., Jacques, J.-E., Roy, V., Lecaille, F., Warszycki, D., Bojarski, A.J., Lalmanach, G., Agrofoglio, L.A.

DOI: 10.1016/j.bmc.2018.07.032
Date: 2018-01-01

Pyrroloquinoline scaffold-based 5-HT<inf>6</inf>R ligands: Synthesis, quantum chemical and molecular dynamic studies, and influence of nitrogen atom position in the scaffold on affinity

Autorzy: Grychowska, K., Kurczab, R., Śliwa, P., Satała, G., Dubiel, K., Matłoka, M., Moszczyński-Pętkowski, R., Pieczykolan, J., Bojarski, A.J., Zajdel, P.

DOI: 10.1016/j.bmc.2018.05.033
Date: 2018-01-01

The effect of the intramolecular C-H⋯O interactions on the conformational preferences of bis-arylsulfones-5-HT<inf>6</inf>receptor antagonists and beyond

Autorzy: Kalinowska-Tłuścik, J., Staroń, J., Krawczuk, A., Mordalski, S., Warszycki, D., Satała, G., Hogendorf, A.S., Bojarski, A.J.

DOI: 10.1039/c8ra03107j
Date: 2018-01-01

Spiro[pyrrolidine-3,3′-oxindoles] as 5-HT<inf>7</inf>receptor ligands

Autorzy: Kelemen, Á.A., Satała, G., Bojarski, A.J., Keserű, G.M.

DOI: 10.1016/j.bmcl.2018.06.019
Date: 2018-01-01

Novel multi-target azinesulfonamides of cyclic amine derivatives as potential antipsychotics with pro-social and pro-cognitive effects

Autorzy: Zajdel, P., Kos, T., Marciniec, K., Satała, G., Canale, V., Kamiński, K., Hołuj, M., Lenda, T., Koralewski, R., Bednarski, M., Nowiński, L., Wójcikowski, J., Daniel, W.A., Nikiforuk, A., Nalepa, I., Chmielarz, P., Kuśmierczyk, J., Bojarski, A.J., Popik, P.

DOI: 10.1016/j.ejmech.2018.01.002
Date: 2018-01-01

Zobacz także