prof. dr hab. Andrzej Bojarski

prof. dr hab. Andrzej Bojarski

+48 12 6623365
pokój 325
Zakład Chemii Leków

Dokonania naukowe

  • Publikacje

Low-basicity 5-HT<inf>7</inf>Receptor Agonists Synthesized Using the van Leusen Multicomponent Protocol

Autorzy: Hogendorf, A.S., Hogendorf, A., Kurczab, R., Satała, G., Lenda, T., Walczak, M., Latacz, G., Handzlik, J., Kieć-Kononowicz, K., Wierońska, J.M., Woźniak, M., Cieślik, P., Bugno, R., Staroń, J., Bojarski, A.J.

DOI: 10.1038/s41598-017-00822-4
Date: 2017-01-01

Ligand-guided homology modelling of the GABA<inf>B2</inf>subunit of the GABA<inf>B</inf>receptor

Autorzy: Freyd, T., Warszycki, D., Mordalski, S., Bojarski, A.J., Sylte, I., Gabrielsen, M.

DOI: 10.1371/journal.pone.0173889
Date: 2017-01-01

Design, Synthesis and Biological Evaluation of Potent Antioxidant 1-(2,5-Dimethoxybenzyl)-4-arylpiperazines and N-Azolyl Substituted 2-(4-Arylpiperazin-1-yl)

Autorzy: Saadeh, H.A., Khasawneh, M.A., Samadi, A., El-Haty, I.A., Satała, G., Bojarski, A.J., Ismaili, L., Bautista-Aguilera, Ó.M., Yañez, M., Mestres, J., Marco-Contelles, J.

DOI: 10.1002/slct.201700397
Date: 2017-01-01

Novel 5-HT<inf>7</inf>R antagonists, arylsulfonamide derivatives of (aryloxy)propyl piperidines: Add-on effect to the antidepressant activity of SSRI and DRI, and pro-cognitive profile

Autorzy: Canale, V., Partyka, A., Kurczab, R., Krawczyk, M., Kos, T., Satała, G., Kubica, B., Jastrzębska-Więsek, M., Wesołowska, A., Bojarski, A.J., Popik, P., Zajdel, P.

DOI: 10.1016/j.bmc.2017.03.057
Date: 2017-01-01

Quo vadis G protein-coupled receptor ligands? A tool for analysis of the emergence of new groups of compounds over time

Autorzy: Leśniak, D., Jastrzębski, S., Podlewska, S., Czarnecki, W.M., Bojarski, A.J.

DOI: 10.1016/j.bmcl.2016.12.001
Date: 2017-01-01

Serotonin transporter and receptor ligands with antidepressant activity as neuroprotective and proapoptotic agents

Autorzy: Chilmonczyk, Z., Bojarski, A.J., Pilc, A., Sylte, I.

DOI: 10.1016/j.pharep.2017.01.011
Date: 2017-01-01

The impact of the halogen bonding on D<inf>2</inf>and 5-HT<inf>1A</inf>/5-HT<inf>7</inf>receptor activity of azinesulfonamides of 4-[(2-ethyl)piperidinyl-1-yl]phenylpiperazines with antipsychotic and antidepressant properties

Autorzy: Partyka, A., Kurczab, R., Canale, V., Satała, G., Marciniec, K., Pasierb, A., Jastrzębska-Więsek, M., Pawłowski, M., Wesołowska, A., Bojarski, A.J., Zajdel, P.

DOI: 10.1016/j.bmc.2017.04.046
Date: 2017-01-01

An algorithm to identify target-selective ligands - A case study of 5-HT7/5-HT1A receptor selectivity

Autorzy: Kurczab, R., Canale, V., Zajdel, P., Bojarski, A.J.

DOI: 10.1371/journal.pone.0156986
Date: 2016-01-01

Arylpiperazinylalkyl derivatives of 8-amino-1,3-dimethylpurine-2,6-dione as novel multitarget 5-HT/D receptor agents with potential antipsychotic activity

Autorzy: Chłoń-Rzepa, G., Bucki, A., Kołaczkowski, M., Partyka, A., Jastrzębska-Więsek, M., Satała, G., Bojarski, A.J., Kalinowska-Tłuścik, J., Kazek, G., Mordyl, B., Głuch-Lutwin, M., Wesołowska, A.

DOI: 10.3109/14756366.2015.1088844
Date: 2016-01-01

Antidepressant-like activity of aroxyalkyl derivatives of 2-methoxyphenylpiperazine and evidence for the involvement of serotonin receptor subtypes in their mechanism of action

Autorzy: Kubacka, M., Mogilski, S., Bednarski, M., Nowiński, L., Dudek, M., Zmudzka, E., Siwek, A., Waszkielewicz, A.M., Marona, H., Satała, G., Bojarski, A., Filipek, B., Pytka, K.

DOI: 10.1016/j.pbb.2015.11.013
Date: 2016-01-01

Zobacz także