prof. dr hab. Andrzej Bojarski

prof. dr hab. Andrzej Bojarski

+48 12 6623365
pokój 325
Zakład Chemii Leków

Dokonania naukowe

  • Publikacje

SAR-studies on the importance of aromatic ring topologies in search for selective 5-HT<inf>7</inf>receptor ligands among phenylpiperazine hydantoin derivatives

Autorzy: Handzlik, J., Bojarski, A.J., Satała, G., Kubacka, M., Sadek, B., Ashoor, A., Siwek, A., Wiȩcek, M., Kucwaj, K., Filipek, B., Kieć-Kononowicz, K.

DOI: 10.1016/j.ejmech.2014.01.065
Date: 2014-01-01

Ligand-directed trafficking of receptor stimulus

Autorzy: Chilmonczyk, Z., Bojarski, A.J., Sylte, I.

DOI: 10.1016/j.pharep.2014.06.006
Date: 2014-01-01

Quinoline-and isoquinoline-sulfonamide analogs of aripiprazole: Novel antipsychotic agents?

Autorzy: Zajdel, P., Partyka, A., Marciniec, K., Bojarski, A.J., Pawlowski, M., Wesolowska, A.

DOI: 10.4155/fmc.13.158
Date: 2014-01-01

Structure-activity relationships and molecular modeling studies of novel arylpiperazinylalkyl 2-benzoxazolones and 2-benzothiazolones as 5-HT<inf>7</inf>and 5-HT<inf>1A</inf>receptor ligands

Autorzy: Salerno, L., Pittalà, V., Modica, M.N., Siracusa, M.A., Intagliata, S., Cagnotto, A., Salmona, M., Kurczab, R., Bojarski, A.J., Romeo, G.

DOI: 10.1016/j.ejmech.2014.08.023
Date: 2014-01-01

Solid-supported synthesis, molecular modeling, and biological activity of long-chain arylpiperazine derivatives with cyclic amino acid amide fragments as 5-HT<inf>7</inf>and 5-HT<inf>1A</inf>receptor ligands

Autorzy: Canale, V., Guzik, P., Kurczab, R., Verdie, P., Satała, G., Kubica, B., Pawłowski, M., Martinez, J., Subra, G., Bojarski, A.J., Zajdel, P.

DOI: 10.1016/j.ejmech.2014.03.005
Date: 2014-01-01

Synthesis and anticonvulsant activity of N-(trans)- 3-phenylprop-2-en-1-yl (cinnamyl) derivatives of aminoalkanols

Autorzy: Gunia-Krzyzak, A., Waszkielewicz, A.M., Słoczyńska, K., Borczuch-Kostańska, M., Cegła, M., Satała, G., Bojarski, A.J., Marona, H.

DOI: 10.2174/1570180811666140423203639
Date: 2014-01-01

The influence of negative training set size on machine learning-based virtual screening

Autorzy: Kurczab, R., Smusz, S., Bojarski, A.J.

DOI: 10.1186/1758-2946-6-32
Date: 2014-01-01

New 7-arylpiperazinylalkyl-8-morpholin-4-yl-purine-2,6-dione derivatives with anxiolytic activity - Synthesis, crystal structure and structure-activity study

Autorzy: Chłoń-Rzepa, G., Zmudzki, P., Pawłowski, M., Wesołowska, A., Satała, G., Bojarski, A.J., Jabłoński, M., Kalinowska-Tłuścik, J.

DOI: 10.1016/j.molstruc.2014.03.018
Date: 2014-01-01

Synthesis and evaluation of antidepressant-like activity of some 4-substituted 1-(2-methoxyphenyl) piperazine derivatives

Autorzy: Waszkielewicz, A.M., Pytka, K., Rapacz, A., Wełna, E., Jarzyna, M., Satała, G., Bojarski, A., Sapa, J., Zmudzki, P., Filipek, B., Marona, H.

DOI: 10.1111/cbdd.12394
Date: 2014-01-01

New 1-arylindoles based serotonin 5-HT<inf>7</inf>antagonists. Synthesis and binding evaluation studies

Autorzy: Sagnes, C., Fournet, G., Satala, G., Bojarski, A.J., Joseph, B.

DOI: 10.1016/j.ejmech.2014.01.055
Date: 2014-01-01

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