prof. dr hab. Andrzej Bojarski
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prof. dr hab. Andrzej Bojarski

prof. dr hab. Andrzej Bojarski
Dokonania naukowe
- Publikacje
Sulfonamides with the N-alkyl-N′-dialkylguanidine moiety as 5-HT<inf>7</inf>receptor ligands
Autorzy: Zajdel, P., Subra, G., Verdie, P., Gabzdyl, E., Bojarski, A.J., Duszyńska, B., Martinez, J., Pawłowski, M.
DOI: 10.1016/j.bmcl.2009.06.038
Date: 2009-01-01
The influence of an ethylene spacer on the 5-HT<inf>1A</inf>and 5-HT<inf>2A</inf>receptor affinity of arylpiperazine derivatives of amides with N-acylated amino acids and 3-differently substituted pyrrolidine-2,5-diones
Autorzy: Zajdel, P., Subra, G., Verdie, P., Bojarski, A.J., Duszyńska, B., Basista, K., Obniska, J., Martinez, J., Pawłowski, M.
DOI: 10.1016/j.ejmech.2008.05.021
Date: 2009-01-01
Synthesis and serotonin receptor activity of the arylpiperazine alkyl/propoxy derivatives of new azatricycloundecanes
Autorzy: Bojarski, A.J., Kuran, B., Kossakowski, J., Kozioł, A., Jagiełło-Wójtowicz, E., Chodkowska, A.
DOI: 10.1016/j.ejmech.2008.03.019
Date: 2009-01-01
Synthesis of 4-substituted 2-(4-methylpiperazino)pyrimidines and quinazoline analogs as serotonin 5-HT<inf>2A</inf>receptor ligands
Autorzy: Saczewski, J., Paluchowska, A., Klenc, J., Raux, E., Barnes, S., Sullivan, S., Duszynska, B., Bojarski, A.J., Strekowskia, L.
DOI: 10.1002/jhet.236
Date: 2009-01-01
Atomic diversity, molecular diversity, and chemical diversity: The concept of chemodiversity
Autorzy: Testa, B., Vistoli, G., Pedretti, A., Bojarski, A.J.
DOI: 10.1002/cbdv.200900071
Date: 2009-01-01
The synthesis of cyclic and acyclic long-chain arylpiperazine derivatives of salicylamide as serotonin receptor ligands
Autorzy: Kowalski, P., Jaśkowska, J., Bojarski, A.J., Duszyńska, B.
DOI: 10.1002/jhet.5570450125
Date: 2008-01-01
Synthesis of new arylpiperazinylalkylthiobenzimidazole, benzothiazole, or benzoxazole derivatives as potent and selective 5-HT<inf>1A</inf> serotonin receptor ligands
Autorzy: Siracusa, M.A., Salerno, L., Modica, M.N., Pittalà, V., Romeo, G., Amato, M.E., Nowak, M., Bojarski, A.J., Mereghetti, I., Cagnotto, A., Mennini, T.
DOI: 10.1021/jm800176x
Date: 2008-01-01
Synthesis and biological properties of 1,8-naphthalimidebutylamines. Serotonin 5-HT<inf>1A</inf>and 5-HT<inf>7</inf>binding data and PASS-assisted search
Autorzy: Kowalski, P., Kowalska, T., Bojarski, A.J., Duszyńska, B.
DOI: 10.1002/jhet.5570440423
Date: 2007-01-01
Novel class of arylpiperazines containing N-acylated amino acids: Their synthesis, 5-HT<inf>1A</inf>, 5-HT<inf>2A</inf>receptor affinity, and in vivo pharmacological evaluation
Autorzy: Zajdel, P., Subra, G., Bojarski, A.J., Duszyńska, B., Tatarczyńska, E., Nikiforuk, A., Chojnacka-Wójcik, E., Pawłowski, M., Martinez, J.
DOI: 10.1016/j.bmc.2007.02.018
Date: 2007-01-01
Fujita-Ban QSAR analysis and CoMFA study of quinoline antagonists of immunostimulatory CpG-oligodeoxynucleotides
Autorzy: Paliakov, E., Henary, M., Say, M., Patterson, S.E., Parker, A., Manzel, L., Macfarlane, D.E., Bojarski, A.J., Strekowski, L.
DOI: 10.1016/j.bmc.2006.09.059
Date: 2007-01-01