prof. dr hab. Andrzej Bojarski

prof. dr hab. Andrzej Bojarski

+48 12 6623365
pokój 325
Zakład Chemii Leków

Dokonania naukowe

  • Publikacje

Structure-intrinsic activity relationship studies in the group of 1-imido/amido substituted 4-(4-arylpiperazin-1-yl)cyclohexane derivatives; new, potent 5-HT<inf>1A</inf>receptor agents with anxiolytic-like activity

Autorzy: Bojarski, A.J., Paluchowska, M.H., Duszyńska, B., Bugno, R., Kłodzińska, A., Tatarczyńska, E., Chojnacka-Wójcik, E.

DOI: 10.1016/j.bmc.2005.09.060
Date: 2006-01-01

Synthesis, anticonvulsant activity and 5-HT1A, 5-HT2A receptor affinity of new N-[(4-arylpiperazin-1-yl)-alkyl] derivatives of 2-azaspiro[4.4]nonane and [4.5]decane-1,3-dione

Autorzy: Obniska, J., Kołaczkowski, M., Bojarski, A.J., Duszyńska, B.

DOI: 10.1016/j.ejmech.2006.03.001
Date: 2006-01-01

Arylpiperazines with N-acylated amino acids as 5-HT<inf>1A</inf>receptor ligands

Autorzy: Zajdel, P., Subra, G., Bojarski, A.J., Duszyńska, B., Pawłowski, M., Martinez, J.

DOI: 10.1016/j.bmcl.2006.04.035
Date: 2006-01-01

Synthesis, anticonvulsant properties and 5-HT1A/5-HT2A receptor affinity of new N-[(4-arylpiperazin-1-yl)-propyl]-2-aza-spiro[4.4] nonane and [4.5]decane-1,3-dione derivatives

Autorzy: Obniska, J, Kolaczkowski, M, Charakchieva-Minol, S, Nedza, K, Dybala, M, Bojarski, AJ

DOI:
Date: 2005-01-01

Synthesis, anticonvulsant properties and 5-HT<inf>1A</inf>/5-HT<inf>2A</inf> receptor affinity of new N-[(4-arylpiperazin-1-yl)-propyl]-2-aza-spiro[4.4] nonane and [4.5]decane-1,3-dione derivatives

Autorzy: Obniska, J., Kołaczkowski, M., Charakchieva-Minol, S., Nedza, K., Dybała, M., Bojarski, A.J.

DOI:
Date: 2005-01-01

Parallel solid-phase synthesis and characterization of new sulfonamide and carboxamide proline derivatives as potential CNS agents

Autorzy: Zajdel, P., Subra, G., Bojarski, A.J., Duszyńska, B., Pawłowski, M., Martinez, J.

DOI: 10.1016/j.bmc.2005.01.060
Date: 2005-01-01

1-Aryl-4-(4-succinimidobutyl)piperazines and their conformationally constrained analogues: Synthesis, binding to serotonin (5-HT<inf>1A</inf>, 5-HT<inf>2A</inf>, 5-HT<inf>7</inf>), α<inf>1</inf>-adrenergic, and dopaminergic D<inf>2</inf>receptors, and in vivo 5-HT<inf>1A</inf>functional characteristics

Autorzy: Bojarski, A.J., Paluchowska, M.H., Duszyńska, B., Kłodzińska, A., Tatarczyńska, E., Chojnacka-Wójcik, E.

DOI: 10.1016/j.bmc.2004.12.041
Date: 2005-01-01

Synthesis and 5-HT<inf>1A</inf>, 5-HT<inf>2A</inf>receptor activity of new β-tetralonohydantoins

Autorzy: Byrtus, H., Pawłowski, M., Czopek, A., Bojarski, A.J., Duszyńska, B., Nowak, G., Kłodzińska, A., Tatarczyńska, E., Wesołowska, A., Chojnacka-Wójcik, E.

DOI: 10.1016/j.ejmech.2004.07.013
Date: 2005-01-01

Novel, flexible, and conformationally defined analogs of gepirone: Synthesis and 5-HT<inf>1A</inf>, 5-HT<inf>2A</inf>, and D<inf>2</inf>receptor activity

Autorzy: Paluchowska, M.H., Bugno, R., Bojarski, A.J., Charakchieva-Minol, S., Duszyńska, B., Tatarczyńska, E., Kłodzińska, A., Stachowicz, K., Chojnacka-Wójcik, E.

DOI: 10.1016/j.bmc.2004.11.019
Date: 2005-01-01

Introduction of a new complex imide system into the structure of LCAPs. The synthesis and a 5-HT1A, 5-HT2A and D2 receptor binding study

Autorzy: Kossakowski, J., Raszkiewicz, A., Bugno, R., Bojarski, A.J.

DOI:
Date: 2004-01-01

Zobacz także