prof. dr hab. Andrzej Bojarski

prof. dr hab. Andrzej Bojarski

+48 12 6623365
pokój 325
Zakład Chemii Leków

Dokonania naukowe

  • Publikacje

The searching of novel PAM of mGluR III by Virtual Screening of commercial chemical databases

Autorzy: Kurczab, Rafal, Bojarski, Andrzej J.

DOI: 10.1016/S1734-1140(12)70803-4
Date: 2012-01-01

Quinoline- and isoquinoline-sulfonamide derivatives of LCAP as potent CNS multi-receptor - 5-HT<inf>1A</inf>/5-HT<inf>2A</inf>/5-HT<inf>7</inf>and D<inf>2</inf>/D<inf>3</inf>/D<inf>4</inf>- Agents: The synthesis and pharmacological evaluation

Autorzy: Zajdel, P., Marciniec, K., Maślankiewicz, A., Satała, G., Duszyńska, B., Bojarski, A.J., Partyka, A., Jastrzbska-Wisek, M., Wróbel, D., Wesołowska, A., Pawłowski, M.

DOI: 10.1016/j.bmc.2011.12.039
Date: 2012-01-01

Synthesis, anticonvulsant activity and 5-HT<inf>1A</inf>/5-HT<inf>7</inf>receptors affinity of 1-[(4-arylpiperazin-1-yl)-propyl]-succinimides

Autorzy: Obniska, J., Chlebek, I., Kamiński, K., Bojarski, A.J., Satała, G.

DOI: 10.1016/S1734-1140(12)70772-7
Date: 2012-01-01

Molecular mechanism of serotonin transporter inhibition elucidated by a new flexible docking protocol

Autorzy: Gabrielsen, M., Kurczab, R., Ravna, A.W., Kufareva, I., Abagyan, R., Chilmonczyk, Z., Bojarski, A.J., Sylte, I.

DOI: 10.1016/j.ejmech.2011.09.056
Date: 2012-01-01

The multiobjective based design, synthesis and evaluation of the arylsulfonamide/amide derivatives of aryloxyethyl and arylthioethyl-piperidines and pyrrolidines as a novel class of potent 5-HT<inf>7</inf>receptor antagonists

Autorzy: Zajdel, P., Kurczab, R., Grychowska, K., Satała, G., Pawłowski, M., Bojarski, A.J.

DOI: 10.1016/j.ejmech.2012.07.043
Date: 2012-01-01

Mass-spectrometric studies of new 6-nitroquipazines-serotonin transporter inhibitors

Autorzy: Witowska-Jarosz, J., Jarończyk, M., Mazurek, A.P., Sylte, I., Bojarski, A.J., Chilmonczyk, Z., Jarosz, M.

DOI: 10.1007/s00216-011-5410-8
Date: 2012-01-01

Synthesis, in vitro binding studies and docking of long-chain arylpiperazine nitroquipazine analogues, as potential serotonin transporter inhibitors

Autorzy: Jarończyk, M., Wołosewicz, K., Gabrielsen, M., Nowak, G., Kufareva, I., Mazurek, A.P., Ravna, A.W., Abagyan, R., Bojarski, A.J., Sylte, I., Chilmonczyk, Z.

DOI: 10.1016/j.ejmech.2012.01.012
Date: 2012-01-01

IF270750: Synthesis and pharmacology of novel mGluR<sub>4</sub> positive allosteric modulator

Autorzy: Branski, Piotr, Stankiewicz, Anna, Bojarski, Andrzej, Burnat, Grzegorz, Chorobik, Paulina, Chruscicka, Barbara, Bugno, Ryszard, Palucha-Poniewiera, Agnieszka, Pilc, Andrzej

DOI:
Date: 2012-01-01

Influence of new high affinity serotonin transporter ligands on cellular cAMP levels

Autorzy: Chilmonczyk, Zdzislaw, Kossakowski, Jerzy, Walory, Jaroslaw, Koronkiewicz, Miroslawa, Sylte, Ingebrigt, Nowak, Gabriel, Bojarski, Andrzej J.

DOI: 10.1016/S1734-1140(11)70534-5
Date: 2011-01-01

How to find a needle in a haystack? The application of in silico methods in searching of potentially new PAM of mGluR III

Autorzy: Kurczab, Rafal, Bojarski, Andrzej J.

DOI: 10.1016/S1734-1140(11)70551-5
Date: 2011-01-01

Zobacz także