prof. dr hab. Andrzej Bojarski

prof. dr hab. Andrzej Bojarski

+48 12 6623365
pokój 325
Zakład Chemii Leków

Dokonania naukowe

  • Publikacje

Synthesis and structural investigation of some pyrimido[5,4-c]quinolin- 4(3H)-one derivatives with a long-chain arylpiperazine moiety as potent 5-HT<inf>1A/2A</inf>and 5-HT<inf>7</inf>receptor ligands

Autorzy: Lewgowd, W., Bojarski, A.J., Szczesio, M., Olczak, A., Glowka, M.L., Mordalski, S., Stanczak, A.

DOI: 10.1016/j.ejmech.2011.04.060
Date: 2011-01-01

Synthesis and characterization of novel metabotropic glutamate receptor 2/3 (mGluR<sub>2/3</sub>) positive allosteric modulator (PAM)

Autorzy: Branski, Piotr, Staron, Jakub, Bugno, Ryszard, Wieronska, Joanna, Bojarski, Andrzej, Burnat, Grzegorz, Palucha-Poniewiera, Agnieszka, Pilc, Andrzej

DOI:
Date: 2011-01-01

Screening for new 5HT(1A) receptor agonists and antagonists

Autorzy: Chilmonczyk, Zdzislaw, Mazurek, Andrzej, Plucinski, Franciszek, Mazurek, Aleksander P., Bojarski, Andrzej J.

DOI: 10.1016/S1734-1140(10)71130-0
Date: 2010-01-01

SAR studies on new bis-aryls 5-HT<inf>7</inf> ligands: Synthesis and molecular modeling

Autorzy: Badarau, E., Bugno, R., Suzenet, F., Bojarski, A.J., Finaru, A.-L., Guillaumet, G.

DOI: 10.1016/j.bmc.2010.01.035
Date: 2010-01-01

New insights into homopiperazine-based 5-HT1A/5-HT7R ligands: Synthesis and biological evaluation

Autorzy: Badarau, E., Putey, A., Suzenet, F., Joseph, B., Bojarski, A., Finaru, A., Guillaumet, G.

DOI: 10.3109/14756360903179393
Date: 2010-01-01

The development and validation of a novel virtual screening cascade protocol to identify potential serotonin 5-HT<inf>7</inf>R antagonists

Autorzy: Kurczab, R., Nowak, M., Chilmonczyk, Z., Sylte, I., Bojarski, A.J.

DOI: 10.1016/j.bmcl.2010.03.012
Date: 2010-01-01

Different neurochemical effects of R and S enantiomers of tetrahydroisoquinoline on dopamine metabolism in rat brain

Autorzy: Antkiewicz-Michaluk, L., Romanska, I., Boksa, J., Bojarski, A., Michaluk, J.

DOI: 10.1016/S0924-977X(09)70378-5
Date: 2009-01-01

The comparison of effects of the endogenous enantiomer, (R)- with the racemate (R,S)-1-methyl-1,2,3,4-tetrahydroisoquinoline on dopamine metabolism in the brain structures and its in vivo release in rat striatum

Autorzy: Wasik, Agnieszka, Michaluk, Jerzy, Romanska, Irena, Bojarski, Andrzej, Antkiewicz-Michaluk, Lucyna

DOI:
Date: 2009-01-01

Simulations in evolution. II. Relative fitness and the propagation of mutants

Autorzy: Testa, B., Bojarski, A.J.

DOI: 10.1002/cbdv.200800303
Date: 2009-01-01

Benzimidazolone-based serotonin 5-HT<inf>1A</inf> or 5-HT<inf>7</inf>R ligands: Synthesis and biological evaluation

Autorzy: Badarau, E., Suzenet, F., Bojarski, A.J., Fînaru, A.-L., Guillaumet, G.

DOI: 10.1016/j.bmcl.2009.02.008
Date: 2009-01-01

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