prof. dr hab. Andrzej Bojarski

prof. dr hab. Andrzej Bojarski

+48 12 6623365
pokój 325
Zakład Chemii Leków

Dokonania naukowe

  • Publikacje

Novel D<sub>2</sub>/5-HT receptor modulators related to cariprazine with potential implication to schizophrenia treatment

Autorzy: Juza, Radomir, Vojtechova, Iveta, Stefkova-Mazochova, Kristyna, Dehaen, Wim, Petrasek, Tomas, Prchal, Lukas, Kobrlova, Tereza, Janousek, Jiri, Vlcek, Premysl, Mezeiova, Eva, Svozil, Daniel, Karasova, Jana Zdarova, Pejchal, Jaroslav, Stark, Holger, Satala, Grzegorz J., Bojarski, Andrzej J., Kubacka, Monika, Mogilski, Szczepan, Randakova, Alena, Musilek, Kamil, Soukup, Ondrej, Korabecny, Jan

DOI: 10.1016/J.EJMECH.2022.114193
Date: 2022-01-01

Serodolin, a β-arrestin-biased ligand of 5-HT7 receptor, attenuates pain-related behaviors

Autorzy: El Khamlichi, Chayma, Reverchon, Flora, Hervouet-Coste, Nadege, Robin, Elodie, Chopin, Nicolas, Deau, Emmanuel, Madouri, Fahima, Guimpied, Cyril, Colas, Cyril, Menuet, Arnaud, Inoue, Asuka, Bojarski, Andrzej J., Guillaumet, Gerald, Suzenet, Franck, Reiter, Eric, Morisset-Lopez, Severine

DOI: 10.1073/PNAS.2118847119
Date: 2022-01-01

Overcoming undesirable hERG affinity by incorporating fluorine atoms: A case of MAO-B inhibitors derived from 1 <i>H</i>-pyrrolo-[3,2-<i>c</i>] quinolines

Autorzy: Grychowska, Katarzyna, Olejarz-Maciej, Agnieszka, Blicharz, Klaudia, Pietrus, Wojciech, Karcz, Tadeusz, Kurczab, Rafal, Koczurkiewicz, Paulina, Doroz-Plonka, Agata, Latacz, Gniewomir, Keeri, Abdul Raheem, Piska, Kamil, Satala, Grzegorz, Pegiel, Joanna, Trybala, Wojciech, Jastrzebska-Wiesek, Magdalena, Bojarski, Andrzej J., Lamaty, Frederic, Partyka, Anna, Walczak, Maria, Krawczyk, Martyna, Malikowska-Racia, Natalia, Popik, Piotr, Zajdel, Pawel

DOI: 10.1016/J.EJMECH.2022.114329
Date: 2022-01-01

New 1,2,4-oxadiazole derivatives with positive mGlu<sub>4</sub> receptor modulation activity and antipsychotic-like properties

Autorzy: Stankiewicz, Anna, Kaczorowska, Katarzyna, Bugno, Ryszard, Koziol, Aneta, Paluchowska, Maria H., Burnat, Grzegorz, Chruscicka, Barbara, Chorobik, Paulina, Branski, Piotr, Wieronska, Joanna M., Duszynska, Beata, Pilc, Andrzej, Bojarski, Andrzej J.

DOI: 10.1080/14756366.2021.1998022
Date: 2022-01-01

Structural and Molecular Insight into Piperazine and Piperidine Derivatives as Histamine H<sub>3</sub> and Sigma-1 Receptor Antagonists with Promising Antinociceptive Properties

Autorzy: Szczepanska, Katarzyna, Podlewska, Sabina, Dichiara, Maria, Gentile, Davide, Patamia, Vincenzo, Rosier, Niklas, Moennich, Denise, Ruiz Cantero, Ma Carmen, Karcz, Tadeusz, Lazewska, Dorota, Siwek, Agata, Pockes, Steffen, Cobos, Enrique J., Marrazzo, Agostino, Stark, Holger, Rescifina, Antonio, Bojarski, Andrzej J., Amata, Emanuele, Kiec-Kononowicz, Katarzyna

DOI: 10.1021/ACSCHEMNEURO.1C00435
Date: 2022-01-01

Comparison of an Addictive Potential of μ-Opioid Receptor Agonists with G Protein Bias: Behavioral and Molecular Modeling Studies

Autorzy: Lucja Kudla, Ryszard Bugno, Sabina Podlewska, Lukasz Szumiec, Lucja Wiktorowska, Andrzej Bojarski, Ryszard Przewlocki

DOI: 10.3390/pharmaceutics14010055
Date: 2021-12-01

Data-Driven Analysis of Fluorination of Ligands of Aminergic G Protein Coupled Receptors

Autorzy: Wojciech Pietruś, Rafał Kurczab, Dagmar Stumpfe, Andrzej Bojarski, Jürgen Bajorath

DOI: 10.3390/biom11111647
Date: 2021-11-01

In Search of Effective Anticancer Agents—Novel Sugar Esters Based on Polyhydroxyalkanoate Monomers

Autorzy: Wojciech Snoch, Dawid Wnuk, Tomasz Witko, Jakub Staroń, Andrzej Bojarski, Ewelina Jarek, Francisco J. Plou, Maciej Guzik

DOI: 10.3390/ijms22137238
Date: 2021-07-01

<i>N</i>-Skatyltryptamines—Dual 5-HT<sub>6</sub>R/D<sub>2</sub>R Ligands with Antipsychotic and Procognitive Potential

Autorzy: Agata Hogendorf, Adam Hogendorf, Rafał Kurczab, Grzegorz Satała, Bernadeta Szewczyk, Paulina Cieślik, Gniewomir Latacz, Jadwiga Handzlik, Tomasz Lenda, Katarzyna Kaczorowska, Jakub Staroń, Ryszard Bugno, Beata Duszyńska, Andrzej Bojarski

DOI: 10.3390/molecules26154605
Date: 2021-07-01

Design, synthesis and biological evaluation of 2-substituted-6-[(4-substituted-1-piperidyl)methyl]-1H-benzimidazoles as inhibitors of ebola virus infection

Autorzy: Bessieres, Maxime, Plebanek, Elzbieta, Chatterjee, Payel, Shrivastava-Ranjan, Punya, Flint, Mike, Spiropoulou, Christina F., Warszycki, Dawid, Bojarski, Andrzej J., Roy, Vincent, Agrofoglio, Luigi A.

DOI: 10.1016/J.EJMECH.2021.113211
Date: 2021-01-01

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