prof. dr hab. Andrzej Bojarski
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prof. dr hab. Andrzej Bojarski

prof. dr hab. Andrzej Bojarski
Dokonania naukowe
- Publikacje
Synthesis, in vitro and in vivo 5-HT<inf>1A</inf>/5-HT<inf>2A</inf> serotonin receptor activity of new hybrid 1,2,3,4-tetrahydro-γ-carbolines with 1-(2-methoxyphenyl)piperazine moiety
Autorzy: Boksa, J., Charakchieva-Minol, S., Duszyńska, B., Bugno, R., Kłodzińska, A., Tatarczyńska, E., Chojnacka-Wójcik, E., Bojarski, A.J.
DOI:
Date: 2003-01-01
Preliminary study on application of impregnated synthetic peptide TLC stationary phases for the pre-screening of 5-HT<inf>1A</inf> ligands
Autorzy: Zajdel, P., Bojarski, A.J., Byrtus, H., Chłoń-Rzepa, G., Obniska, J., Chevallet, P., Martinez, J., Pawłowski, M.
DOI: 10.1002/bmc.224
Date: 2003-01-01
Modification of the structure of 4,6-disubstituted 2-(4-alkyl-1-piperazinyl)pyridines: Synthesis and their 5-HT<inf>2A</inf> receptor activity
Autorzy: Paluchowska, M.H., Bojarski, A.J., Bugno, R., Charakchieva-Minol, S., Wesołowska, A.
DOI: 10.1002/ardp.200390006
Date: 2003-01-01
Electrospray mass spectrometric studies of noncovalent complexes of buspirone hydrochloride and other serotonin 5-HT<inf>1A</inf>receptor ligands containing arylpiperazine moieties
Autorzy: Kowalski, P., Suder, P., Kowalska, T., Silberring, J., Duszyńska, B., Bojarski, A.J.
DOI: 10.1002/rcm.1166
Date: 2003-01-01
Synthesis and activity of substituted 2-phenylquinolin-4-amines, antagonists of immunostimulatory CpG-oligodeoxynucleotides
Autorzy: Strekowski, L., Say, M., Henary, M., Ruiz, P., Manzel, L., Macfarlane, D.E., Bojarski, A.J.
DOI: 10.1021/jm020374y
Date: 2003-01-01
Synthesis, <i>in vitro</i> and <i>in vivo</i> 5-HT<sub>1A</sub>/5-HT<sub>2A</sub> serotonin receptor activity of new hybrid 1,2,3,4-tetrahydro-γ-carbolines with 1-(2-methoxyphenyl)piperazine moiety
Autorzy: Boksa, J, Charakchieva-Minol, S, Duszynska, B, Bugno, R, Klodzinska, A, Tatarczynska, E, Chojnacka-Wójcik, E, Bojarski, AJ
DOI:
Date: 2003-01-01
Synthesis and pharmacological evaluation of new arylpiperazines. 3-{4-[4-(3-chlorophenyl)-1-piperazinyl]butyl}-quinazolidin-4-one - A dual serotonin 5-HT<inf>1A</inf>/5-HT<inf>2A</inf> receptor ligand with an anxiolytic-like activity
Autorzy: Bojarski, A.J., Kowalski, P., Kowalska, T., Duszyńska, B., Charakchieva-Minol, S., Tatarczyńska, E., Kłodzińska, A., Chojnacka-Wójcik, E.
DOI: 10.1016/S0968-0896(02)00349-8
Date: 2002-01-01
Active conformation of some arylpiperazine postsynaptic 5-HT<inf>1A</inf>receptor antagonists
Autorzy: Paluchowska, M.H., Bojarski, A.J., Charakchieva-Minol, S., Wesołowska, A.
DOI: 10.1016/S0223-5234(01)01312-5
Date: 2002-01-01
The influence of substitution at aromatic part of 1,2,3,4-tetrahydroisoquinoline on in vitro and in vivo 5-HT<inf>1A</inf>/5-HT<inf>2A</inf>receptor activities of its 1-adamantoyloaminoalkyl derivatives
Autorzy: Bojarski, A.J., Mokrosz, M.J., Minol, S.C., Koziol, A., Wesolowska, A., Tatarczyńska, E., Klodzińska, A., Chojnacka-Wójcik, E.
DOI: 10.1016/S0968-0896(01)00236-X
Date: 2002-01-01
Substituted 2-(1,2,3,4-tetrahydroisoquinoline)-butyl derivatives of azaspiro[4.5]decane-7,9-dione and phthalimide as new 5-HT1A and 5-HT2A receptor ligands
Autorzy: Bojarski, AJ, Misztal, S, Boksa, J, Charakchieva-Minol, S, Wesolowska, A, Tatarczynska, E, Klodzinska, A, Chojnacka-Wojcik, E
DOI:
Date: 2001-01-01