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Department of Medicinal Chemistry
Scientific profile
- Employees
Pracownicy zakładu
Ryszard Bugno, dr
+48 12 6623320
bugno@if-pan.krakow.pl
room 331Rafał Kurczab, dr hab.
+48 12 6623301kurczab@if-pan.krakow.plroom 326Sabina Podlewska, dr hab.
+48 12 6623301smusz@if-pan.krakow.plroom 326Grzegorz Satała, dr
+48 12 6623301satala@if-pan.krakow.plroom 326Katarzyna Szczepańska, dr
+48 12 6623301k.szczep@if-pan.krakow.plroom 326Adam Hogendorf, dr
+48 792287874ahogen@if-pan.krakow.plroom 331Katarzyna Kaczorowska, dr
+48 12 3343720k.kaczor@if-pan.krakow.plroom CEPHARES CF2.15Janusz Malarz, dr
+48 12 6623254malarzj@if-pan.krakow.plroom Radzikowskiego 176Wojciech Pietruś, dr
pietrus@if-pan.krakow.plDawid Warszycki, dr
+48 12 6623301warszyc@if-pan.krakow.plroom 326Aneta Kozioł
+48 12 6623319koziol@if-pan.krakow.plroom 330Krystyna Nędza
+48 12 6623319nedza@if-pan.krakow.plroom 330Achievements
- Publications
- Grants
Grant
Development of protocol for in silico design of compounds inhibit Ebola virus infection
Dawid Warszycki, PhD
Quo vadis G protein-coupled receptor ligands? A tool for analysis of the emergence of new groups of compounds over time
Leśniak, D., Jastrzębski, S., Podlewska, S., Czarnecki, W.M., Bojarski, A.J.
DOI: 10.1016/j.bmcl.2016.12.001
Serotonin transporter and receptor ligands with antidepressant activity as neuroprotective and proapoptotic agents
Chilmonczyk, Z., Bojarski, A.J., Pilc, A., Sylte, I.
DOI: 10.1016/j.pharep.2017.01.011
The impact of the halogen bonding on D<inf>2</inf>and 5-HT<inf>1A</inf>/5-HT<inf>7</inf>receptor activity of azinesulfonamides of 4-[(2-ethyl)piperidinyl-1-yl]phenylpiperazines with antipsychotic and antidepressant properties
Partyka, A., Kurczab, R., Canale, V., Satała, G., Marciniec, K., Pasierb, A., Jastrzębska-Więsek, M., Pawłowski, M., Wesołowska, A., Bojarski, A.J., Zajdel, P.
DOI: 10.1016/j.bmc.2017.04.046
Towards new 5-HT<inf>7</inf> antagonists among arylsulfonamide derivatives of (aryloxy)ethyl-alkyl amines: Multiobjective based design, synthesis, and antidepressant and anxiolytic properties
Canale, V., Kurczab, R., Partyka, A., Sataa, G., Ledna, T., Jastrzebska-Wiesek, M., Wesoowska, A., Bojarski, A.J., Zajdel, P.
DOI: 10.1016/j.ejmech.2015.11.040
N-Alkylated arylsulfonamides of (aryloxy)ethyl piperidines: 5-HT<inf>7</inf> receptor selectivity versus multireceptor profile
Canale, V., Kurczab, R., Partyka, A., Satała, G., Słoczyńska, K., Kos, T., Jastrzębska-Więsek, M., Siwek, A., Pękala, E., Bojarski, A.J., Wesołowska, A., Popik, P., Zajdel, P.
DOI: 10.1016/j.bmc.2015.11.041
An algorithm to identify target-selective ligands - A case study of 5-HT7/5-HT1A receptor selectivity
Kurczab, R., Canale, V., Zajdel, P., Bojarski, A.J.
DOI: 10.1371/journal.pone.0156986
Halogen bonding enhances activity in a series of dual 5-HT<inf>6</inf>/D<inf>2</inf> ligands designed in a hybrid bioisostere generation/virtual screening protocol
Staroń, J., Warszycki, D., Kurczab, R., Satała, G., Bugno, R., Hogendorf, A., Bojarski, A.J.
DOI: 10.1039/c6ra08714k
An algorithm to identify target-selective ligands - A case study of 5-HT7/5-HT1A receptor selectivity
Kurczab, R., Canale, V., Zajdel, P., Bojarski, A.J.
DOI: 10.1371/journal.pone.0156986
Arylpiperazinylalkyl derivatives of 8-amino-1,3-dimethylpurine-2,6-dione as novel multitarget 5-HT/D receptor agents with potential antipsychotic activity
Chłoń-Rzepa, G., Bucki, A., Kołaczkowski, M., Partyka, A., Jastrzębska-Więsek, M., Satała, G., Bojarski, A.J., Kalinowska-Tłuścik, J., Kazek, G., Mordyl, B., Głuch-Lutwin, M., Wesołowska, A.
DOI: 10.3109/14756366.2015.1088844
Antidepressant-like activity of aroxyalkyl derivatives of 2-methoxyphenylpiperazine and evidence for the involvement of serotonin receptor subtypes in their mechanism of action
Kubacka, M., Mogilski, S., Bednarski, M., Nowiński, L., Dudek, M., Zmudzka, E., Siwek, A., Waszkielewicz, A.M., Marona, H., Satała, G., Bojarski, A., Filipek, B., Pytka, K.
DOI: 10.1016/j.pbb.2015.11.013