Department of Medicinal Chemistry
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Department of Medicinal Chemistry

Scientific profile
- Employees
Pracownicy zakładu
Ryszard Bugno, dr
Rafał Kurczab, dr hab.
Sabina Podlewska, dr hab.
Grzegorz Satała, dr
Katarzyna Szczepańska, dr
Adam Hogendorf, dr
Katarzyna Kaczorowska, dr
Janusz Malarz, dr
Wojciech Pietruś, dr
Dawid Warszycki, dr
Aneta Kozioł
Krystyna Nędza
Achievements
- Publications
- Grants
Grant
Development of protocol for in silico design of compounds inhibit Ebola virus infection
Dawid Warszycki, PhD
The influence of the inactives subset generation on the performance of machine learning methods
Smusz, S., Kurczab, R., Bojarski, A.J.
DOI: 10.1186/1758-2946-5-17
New strategy for receptor-based pharmacophore query construction: A case study for 5-HT<inf>7</inf> receptor ligands
Kurczab, R., Bojarski, A.J.
DOI: 10.1021/ci4005207
Evaluation of [F-18]MNI-709 and [F-18]MNI-711 as potential 5HT(7) PET imaging agents
Alagille, David, Barret, Olivier, Caille, Fabien, Morisset-Lopez, S., Bojarski, A. J., Finaru, A. L., Suzenet, F., Guillaumet, Gerald, Papin, Caroline, Morley, Tomas, Lee, Sharon, Tavares, Adriana, Seibyl, John, Tamagnan, Gilles
DOI:
Anticonvulsant Activity and 5-HT1A/5-HT7 Receptors Affinity of Piperazine Derivatives of 3,3-Diphenyl- and 3,3-Dimethyl-succinimides
Obniska, Jolanta, Chlebek, Iwona, Kaminski, Krzysztof, Bojarski, Andrzej J., Satala, Grzegorz
DOI: 10.2174/157018013804725116
Anticonvulsant activity and 5-HT1A/5-HT7 receptors affinity of piperazine derivatives of 3,3-diphenyl- and 3,3-dimethyl- succinimides
Obniska, J., Chlebek, I., Kamiński, K., Bojarski, A.J., Satała, G.
DOI:
The influence of the inactives subset generation on the performance of machine learning methods
Smusz, S., Kurczab, R., Bojarski, A.J.
DOI: 10.1186/1758-2946-5-17
New arylpiperazines with flexible versus partly constrained linker as serotonin 5-HT<inf>1A</inf>/5-HT<inf>7</inf> receptor ligands
Kowalski, P., Mitka, K., Jaśkowska, J., Duszyńska, B., Bojarski, A.J.
DOI: 10.1002/ardp.201300011
Simulations in evolution. III. Randomness as a generator of opportunities
Testa, B., Bojarski, A.J., Mordalski, S.
DOI: 10.1002/cbdv.201200207
Antidepressant and antipsychotic activity of new quinoline- and isoquinoline-sulfonamide analogs of aripiprazole targeting serotonin 5-HT 1A/5-HT2A/5-HT7 and dopamine D 2/D3 receptors
Zajdel, P., Marciniec, K., Maślankiewicz, A., Grychowska, K., Satała, G., Duszyńska, B., Lenda, T., Siwek, A., Nowak, G., Partyka, A., Wróbel, D., Jastrzȩbska-Wiȩsek, M., Bojarski, A.J., Wesołowska, A., Pawłowski, M.
DOI: 10.1016/j.ejmech.2012.11.042
Towards metabolically stable 5-HT7 receptor ligands: A study on 1-arylpiperazine derivatives and related isosters
Lacivita, E., De Giorgio, P., Patarnello, D., Niso, M., Colabufo, N.A., Berardi, F., Perrone, R., Satala, G., Duszynska, B., Bojarski, A.J., Leopoldo, M.
DOI: 10.1007/s00221-013-3498-0