Department of Medicinal Chemistry
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Department of Medicinal Chemistry

Scientific profile
- Employees
Pracownicy zakładu
Ryszard Bugno, dr
Rafał Kurczab, dr hab.
Sabina Podlewska, dr hab.
Grzegorz Satała, dr
Katarzyna Szczepańska, dr
Adam Hogendorf, dr
Katarzyna Kaczorowska, dr
Janusz Malarz, dr
Wojciech Pietruś, dr
Dawid Warszycki, dr
Aneta Kozioł
Krystyna Nędza
Achievements
- Publications
- Grants
Grant
Development of protocol for in silico design of compounds inhibit Ebola virus infection
Dawid Warszycki, PhD
Studies on the syntheses of 1-substituted benzimidazole derivatives
Kowalska, T., Kowalski, P., Bojarski, A.J., Duszyńska, B.
DOI:
Protective effect of 1-methyl-1,2,3,4-tetrahydroisoquinoline against dopaminergic neurodegeneration in the extrapyramidal structures produced by intracerebral injection of rotenone
Antkiewicz-Michaluk, L., Wardas, J., Michaluk, J., Romańska, I., Bojarski, A., Vetulani, J.
DOI: 10.1017/S1461145703004036
New Arylpiperazine 5-HT<inf>1A</inf> Receptor Ligands Containing the Pyrimido[2,1-f]purine Fragment: Synthesis, in Vitro, and in Vivo Pharmacological Evaluation
Jurczyk, Sł., Kołaczkowski, M., Maryniak, E., Zajdel, P., Pawłowski, M., Tatarczyńska, E., Kłodzińska, A., Chojnacka-Wójcik, E., Bojarski, A.J., Charakchieva-Minol, S., Duszyńska, B., Nowak, G., Macia̧g, D.
DOI: 10.1021/jm030946u
A study on application of impregnated synthetic peptide TLC stationary phases for the screening of 5-HT<inf>1A</inf> ligands. Part 2
Zajdel, P., Bojarski, A.J., Bugno, R., Jurczyk, S., Kołaczkowski, M., Nowak, M., Subra, G., Martinez, J., Pawłowski, M.
DOI: 10.1002/bmc.354
A new class of arylpiperazine derivatives: The library synthesis on SynPhase Lanterns and biological evaluation on serotonin 5-HT<inf>1A</inf> and 5-HT<inf>2A</inf> receptors
Zajdel, P., Subra, G., Bojarski, A.J., Duszyńska, B., Pawłowski, M., Martinez, J.
DOI: 10.1021/cc049970z
The impact of spacer structure on 5-HT<inf>7</inf>and 5-HT<inf>1A</inf>receptor affinity in the group of long-chain arylpiperazine ligands
Bojarski, A.J., Duszyńska, B., Kołaczkowski, M., Kowalski, P., Kowalska, T.
DOI: 10.1016/j.bmcl.2004.09.029
New imide 5-HT<inf>1A</inf>receptor ligands - Modification of terminal fragment geometry
Bojarski, A.J., Mokrosz, M.J., Duszyńska, B., Kozioł, A., Bugno, R.
DOI: 10.3390/90300170
Introduction of a new complex imide system into the structure of LCAPs.: The synthesis and a 5-HT<sub>1A</sub>, 5-HT<sub>2A</sub> and D<sub>2</sub> receptor binding study
Kossakowski, J, Raszkiewicz, A, Bugno, R, Bojarski, AJ
DOI:
1-Methyl-1,2,3,4-tetrahydroisoquinoline protects against rotenone-induced mortality and biochemical changes in rat brain
Antkiewicz-Michaluk, L., Karolewicz, B., Romańska, I., Michaluk, J., Bojarski, A.J., Vetulani, J.
DOI: 10.1016/S0014-2999(03)01565-6
Conformational constraints on side chains in protein residues increase their information content
Bojarski, A.J., Nowak, M., Testa, B.
DOI: 10.1007/s00018-003-3280-8