Achievements

  • Publications
  • Grants

Grant

Development of protocol for in silico design of compounds inhibit Ebola virus infection

Dawid Warszycki, PhD

Mass-spectrometric studies of new 6-nitroquipazines-serotonin transporter inhibitors

Witowska-Jarosz, J., Jarończyk, M., Mazurek, A.P., Sylte, I., Bojarski, A.J., Chilmonczyk, Z., Jarosz, M.

DOI: 10.1007/s00216-011-5410-8

Synthesis, in vitro binding studies and docking of long-chain arylpiperazine nitroquipazine analogues, as potential serotonin transporter inhibitors

Jarończyk, M., Wołosewicz, K., Gabrielsen, M., Nowak, G., Kufareva, I., Mazurek, A.P., Ravna, A.W., Abagyan, R., Bojarski, A.J., Sylte, I., Chilmonczyk, Z.

DOI: 10.1016/j.ejmech.2012.01.012

IF270750: Synthesis and pharmacology of novel mGluR<sub>4</sub> positive allosteric modulator

Branski, Piotr, Stankiewicz, Anna, Bojarski, Andrzej, Burnat, Grzegorz, Chorobik, Paulina, Chruscicka, Barbara, Bugno, Ryszard, Palucha-Poniewiera, Agnieszka, Pilc, Andrzej

DOI:

Evaluation of different machine learning methods for ligand-based virtual screening

Kurczab, R., Smusz, S., Bojarski, A.J.

DOI: 10.1186/1758-2946-3-S1-P41

Influence of new high affinity serotonin transporter ligands on cellular cAMP levels

Chilmonczyk, Zdzislaw, Kossakowski, Jerzy, Walory, Jaroslaw, Koronkiewicz, Miroslawa, Sylte, Ingebrigt, Nowak, Gabriel, Bojarski, Andrzej J.

DOI: 10.1016/S1734-1140(11)70534-5

Evaluation of 1-arylpiperazine derivative of hydroxybenzamides as 5-HT 1A and 5-HT7 serotonin receptor ligands: An experimental and molecular modeling approach

Kowalski, P., Jaśkowska, J., Bojarski, A.J., Duszyåska, B., Bucki, A., Koåaczkowski, M.

DOI: 10.1002/jhet.526

Evaluation of different machine learning methods for ligand-based virtual screening

Kurczab, R., Smusz, S., Bojarski, A.J.

DOI: 10.1186/1758-2946-3-S1-P41

See also