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Department of Medicinal Chemistry
Scientific profile
- Employees
Pracownicy zakładu
Ryszard Bugno, dr
+48 12 6623320
bugno@if-pan.krakow.pl
room 331Rafał Kurczab, dr hab.
+48 12 6623301kurczab@if-pan.krakow.plroom 326Sabina Podlewska, dr hab.
+48 12 6623301smusz@if-pan.krakow.plroom 326Grzegorz Satała, dr
+48 12 6623301satala@if-pan.krakow.plroom 326Katarzyna Szczepańska, dr
+48 12 6623301k.szczep@if-pan.krakow.plroom 326Adam Hogendorf, dr
+48 792287874ahogen@if-pan.krakow.plroom 331Katarzyna Kaczorowska, dr
+48 12 3343720k.kaczor@if-pan.krakow.plroom CEPHARES CF2.15Janusz Malarz, dr
+48 12 6623254malarzj@if-pan.krakow.plroom Radzikowskiego 176Wojciech Pietruś, dr
pietrus@if-pan.krakow.plDawid Warszycki, dr
+48 12 6623301warszyc@if-pan.krakow.plroom 326Aneta Kozioł
+48 12 6623319koziol@if-pan.krakow.plroom 330Krystyna Nędza
+48 12 6623319nedza@if-pan.krakow.plroom 330Achievements
- Publications
- Grants
Grant
Development of protocol for in silico design of compounds inhibit Ebola virus infection
Dawid Warszycki, PhD
Low-basicity 5-HT<inf>7</inf> Receptor Agonists Synthesized Using the van Leusen Multicomponent Protocol
Hogendorf, A.S., Hogendorf, A., Kurczab, R., Satała, G., Lenda, T., Walczak, M., Latacz, G., Handzlik, J., Kieć-Kononowicz, K., Wierońska, J.M., Woźniak, M., Cieślik, P., Bugno, R., Staroń, J., Bojarski, A.J.
DOI: 10.1038/s41598-017-00822-4
The impact of the halogen bonding on D<inf>2</inf> and 5-HT<inf>1A</inf>/5-HT<inf>7</inf> receptor activity of azinesulfonamides of 4-[(2-ethyl)piperidinyl-1-yl]phenylpiperazines with antipsychotic and antidepressant properties
Partyka, A., Kurczab, R., Canale, V., Satała, G., Marciniec, K., Pasierb, A., Jastrzębska-Więsek, M., Pawłowski, M., Wesołowska, A., Bojarski, A.J., Zajdel, P.
DOI: 10.1016/j.bmc.2017.04.046
Reaction mechanism of sterol hydroxylation by steroid C25 dehydrogenase – Homology model, reactivity and isoenzymatic diversity
Rugor, A., Wójcik-Augustyn, A., Niedzialkowska, E., Mordalski, S., Staroń, J., Bojarski, A., Szaleniec, M.
DOI: 10.1016/j.jinorgbio.2017.04.027
The influence of the negative-positive ratio and screening database size on the performance of machine learning-based virtual screening
Kurczab, R., Bojarski, A.J.
DOI: 10.1371/journal.pone.0175410
Pyrano[2,3,4-cd]indole as a Scaffold for Selective Nonbasic 5-HT<inf>6</inf>R Ligands
Staroń, J., Mordalski, S., Warszycki, D., Satała, G., Hogendorf, A., Bojarski, A.J.
DOI: 10.1021/acsmedchemlett.6b00482
Spiro[pyrrolidine-3, 3′-oxindoles] and their indoline analogues as new 5-HT6 receptor chemotypes
Kelemen, Á.A., Satala, G., Bojarski, A.J., Keseru, G.M.
DOI: 10.3390/molecules22122221
Low-basicity 5-HT<inf>7</inf>Receptor Agonists Synthesized Using the van Leusen Multicomponent Protocol
Hogendorf, A.S., Hogendorf, A., Kurczab, R., Satała, G., Lenda, T., Walczak, M., Latacz, G., Handzlik, J., Kieć-Kononowicz, K., Wierońska, J.M., Woźniak, M., Cieślik, P., Bugno, R., Staroń, J., Bojarski, A.J.
DOI: 10.1038/s41598-017-00822-4
Ligand-guided homology modelling of the GABA<inf>B2</inf>subunit of the GABA<inf>B</inf>receptor
Freyd, T., Warszycki, D., Mordalski, S., Bojarski, A.J., Sylte, I., Gabrielsen, M.
DOI: 10.1371/journal.pone.0173889
Design, Synthesis and Biological Evaluation of Potent Antioxidant 1-(2,5-Dimethoxybenzyl)-4-arylpiperazines and N-Azolyl Substituted 2-(4-Arylpiperazin-1-yl)
Saadeh, H.A., Khasawneh, M.A., Samadi, A., El-Haty, I.A., Satała, G., Bojarski, A.J., Ismaili, L., Bautista-Aguilera, Ó.M., Yañez, M., Mestres, J., Marco-Contelles, J.
DOI: 10.1002/slct.201700397
Novel 5-HT<inf>7</inf>R antagonists, arylsulfonamide derivatives of (aryloxy)propyl piperidines: Add-on effect to the antidepressant activity of SSRI and DRI, and pro-cognitive profile
Canale, V., Partyka, A., Kurczab, R., Krawczyk, M., Kos, T., Satała, G., Kubica, B., Jastrzębska-Więsek, M., Wesołowska, A., Bojarski, A.J., Popik, P., Zajdel, P.
DOI: 10.1016/j.bmc.2017.03.057