Department of Medicinal Chemistry
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Department of Medicinal Chemistry

Scientific profile
- Employees
Pracownicy zakładu
Ryszard Bugno, dr
Rafał Kurczab, dr hab.
Sabina Podlewska, dr hab.
Grzegorz Satała, dr
Katarzyna Szczepańska, dr
Adam Hogendorf, dr
Katarzyna Kaczorowska, dr
Janusz Malarz, dr
Wojciech Pietruś, dr
Dawid Warszycki, dr
Aneta Kozioł
Krystyna Nędza
Achievements
- Publications
- Grants
Grant
Development of protocol for in silico design of compounds inhibit Ebola virus infection
Dawid Warszycki, PhD
Variation, natural selection, and information content - A simulation
Testa, B., Bojarski, A.J.
DOI: 10.1002/cbdv.200790200
7-Arylpiperazinylalkyl and 7-tetrahydroisoquinolinylalkyl derivatives of 8-alkoxy-purine-2,6-dione and some of their purine-2,6,8-trione analogs as 5-HT1A, 5-HT2A, and 5-HT7 serotonin receptor ligands
Chłoń-Rzepa, G., Zmudzki, P., Zajdel, P., Bojarski, A.J., Duszyńska, B., Nikiforuk, A., Tatarczyńska, E., Pawłowski, M.
DOI: 10.1016/j.bmc.2007.05.017
N-acylated amino acid derivatives as serotoninergic receptor ligands
Zajdel, P., Subra, G., Bojarski, A. J., Duszynska, B., Tatarczynska, E., Chojnacka-Wojcik, E., Pawlowski, M., Martinez, J.
DOI:
Antagonists of immunostimulatory CpG-DNA
Paliakov, Ekaterina M., Say, Martial, Henary, Maged M., Macfarlane, Donald, Manzel, Lori, Patterson, Steven E., Bojarski, Andrzej J., Strekowski, Lucjan
DOI:
Structure-activity relationships and modeling studies in the group of 2-(4-methylpiperazino) pyridines as serotonin receptor agents
Raszkiewicz, Aldona, Duszynska, Beata, Bojarski, Andrzej J., Paluchowska, Maria H., Nowak, Mateusz, Kolaczkowski, Marcin, Germann, Markus W., Strekowski, Lucjan
DOI:
Pharmacophore models for metabotropic 5-HT receptor ligands
Bojarski, A.J.
DOI: 10.2174/156802606778522186
Homology modeling of the serotonin 5-HT<inf>1A</inf> receptor using automated docking of bioactive compounds with defined geometry
Nowak, M., Kołaczkowski, M., Pawłowski, M., Bojarski, A.J.
DOI: 10.1021/jm050826h
Conformational fluctuations versus constraints in amino acid side chains: The evolution of information content from free amino acids to proteins
Bojarski, A.J., Nowak, M., Testa, B.
DOI: 10.1002/cbdv.200690029
Conformational restriction in novel NAN-190 and MP3022 analogs and their 5-HT<inf>1A</inf> receptor activity
Paluchowska, M.H., Bugno, R., Charakchieva-Minol, S., Bojarski, A.J., Tatarczyńska, E., Chojnacka-Wójcik, E.
DOI: 10.1002/ardp.200600009
Receptor-based pharmacophores for serotonin 5-HT<inf>7</inf>R antagonists - Implications to selectivity
Kołaczkowski, M., Nowak, M., Pawłowski, M., Bojarski, A.J.
DOI: 10.1021/jm060300c