Achievements

  • Publications
  • Grants

Grant

Development of protocol for in silico design of compounds inhibit Ebola virus infection

Dawid Warszycki, PhD

Solid-Supported Synthesis and 5-HT<inf>7</inf>/5-HT<inf>1A</inf> Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1H)-one

Grychowska, K., Masurier, N., Verdié, P., Satała, G., Bojarski, A.J., Martinez, J., Pawłowski, M., Subra, G., Zajdel, P.

DOI: 10.1111/cbdd.12539

Structure-5-HT Receptor Affinity Relationship in a New Group of 7-Arylpiperazynylalkyl and 7-Tetrahydroisoquinolinylalkyl Derivatives of 8-Amino-1,3-dimethyl-1H-purine-2,6(3H,7H)-dione

Zmudzki, P., Chłoń-Rzepa, G., Bojarski, A.J., Zygmunt, M., Kazek, G., Mordyl, B., Pawłowski, M.

DOI: 10.1002/ardp.201400392

Structure-activity relationships and molecular studies of novel arylpiperazinylalkyl purine-2,4-diones and purine-2,4,8-triones with antidepressant and anxiolytic-like activity

Zagórska, A., Kolaczkowski, M., Bucki, A., Siwek, A., Kazek, G., Satala, G., Bojarski, A.J., Partyka, A., Wesolowska, A., Pawlowski, M.

DOI: 10.1016/j.ejmech.2015.04.046

A new crystal structure fragment-based pharmacophore method for G protein-coupled receptors

Fidom, K., Isberg, V., Hauser, A.S., Mordalski, S., Lehto, T., Bojarski, A.J., Gloriam, D.E.

DOI: 10.1016/j.ymeth.2014.09.009

Rational Design, Pharmacomodulation, and Synthesis of Dual 5-Hydroxytryptamine 7 (5-HT<inf>7</inf>)/5-Hydroxytryptamine 2A (5-HT<inf>2A</inf>) Receptor Antagonists and Evaluation by [<sup>18</sup>F]-PET Imaging in a Primate Brain

Deau, E., Robin, E., Voinea, R., Percina, N., Satała, G., Finaru, A.-L., Chartier, A., Tamagnan, G., Alagille, D., Bojarski, A.J., Morisset-Lopez, S., Suzenet, F., Guillaumet, G.

DOI: 10.1021/acs.jmedchem.5b00874

Novel spirohydantoin derivative as a potent multireceptor-active antipsychotic and antidepressant agent

Czopek, A., Kołaczkowski, M., Bucki, A., Byrtus, H., Pawłowski, M., Kazek, G., Bojarski, A.J., Piaskowska, A., Kalinowska-Tłücik, J., Partyka, A., Wesołowska, A.

DOI: 10.1016/j.bmc.2015.04.026

New Arylpiperazinylalkyl Derivatives of 8-Alkoxy-purine-2,6-dione and Dihydro[1,3]oxazolo[2,3-f]purinedione Targeting the Serotonin 5-HT<inf>1A</inf>/5-HT<inf>2A</inf>/5-HT<inf>7</inf> and Dopamine D<inf>2</inf> Receptors

Chłoń-Rzepa, G., Zagórska, A., Bucki, A., Kołaczkowski, M., Pawłowski, M., Satała, G., Bojarski, A.J., Partyka, A., Wesołowska, A., Pȩkala, E., Słoczyńska, K.

DOI: 10.1002/ardp.201500015

Synthesis of Some Aminophosphonates Bearing N-(Fluorophenyl)-piperazynyl Moiety and Their Activity toward Serotonin Receptors

Lewkowski, J., Jóźwiak, A., Tokarz, P., Zagórski, P.M., Hamera, R., Cal, D., Satała, G., Bojarski, A.J.

DOI: 10.1002/hc.21259

Bioisosteric matrices for ligands of serotonin receptors

Warszycki, D., Mordalski, S., Staroń, J., Bojarski, A.J.

DOI: 10.1002/cmdc.201402563

Robust optimization of SVM hyperparameters in the classification of bioactive compounds

Czarnecki, W.M., Podlewska, S., Bojarski, A.J.

DOI: 10.1186/s13321-015-0088-0

See also