Department of Medicinal Chemistry
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Department of Medicinal Chemistry

Scientific profile
- Employees
Pracownicy zakładu
Ryszard Bugno, dr
Rafał Kurczab, dr hab.
Sabina Podlewska, dr hab.
Grzegorz Satała, dr
Katarzyna Szczepańska, dr
Adam Hogendorf, dr
Katarzyna Kaczorowska, dr
Janusz Malarz, dr
Wojciech Pietruś, dr
Dawid Warszycki, dr
Aneta Kozioł
Krystyna Nędza
Achievements
- Publications
- Grants
Grant
Development of protocol for in silico design of compounds inhibit Ebola virus infection
Dawid Warszycki, PhD
New 9- or 10-arylpiperazinoalkyl substituted pyrimido- or diazepino[2,1- f]purines with partial or full 5-HT(1A) agonistic activity
Pawlowski, M., Katlabi, J., Drabczynska, A., Duszynska, B., Charakchieva-Minol, S., Deren-Wesolek, A., Tatarczynska, E., Chojnacka-Wójcik, E., Mokrosz, M.J., Bojarski, A.J.
DOI: 10.1016/S0223-5234(99)80050-6
On the bioactive conformation of NAN-190 (1) and MP3022 (2), 5-HT(1A) receptor antagonists
Paluchowska, M.H., Mokrosz, M.J., Bojarski, A., Wesołowska, A., Borycz, J., Charakchieva-Minol, S., Chojnacka-Wójcik, E.
DOI: 10.1021/jm991045h
Novel 1,4-benzoxazin-3(4H)-one, 1,2-benzoxazolin-3-one and 1,3- benzoxazolin-2,4-dione arylpiperazine derivatives with different 5-HT(1A) and antagonistic 5-HT(2A) activities
Mokrosz, M.J., Kowalski, P., Kowalska, T., Majka, Z., Duszyńska, B., Bojarski, A.J., Fruziński, A., Karolak-Wojciechowska, J., Wesołowska, A., Kłodzińska, A., Tatarczyńska, E., Chojnacka-Wójcik, E.
DOI: 10.1002/(SICI)1521-4184(199911)332:11<373::AID-ARDP373>3.0.CO;2-L
1,2,3,4-Tetrahydroisoquinoline derivatives: A new class of 5-HT(1A) receptor ligands
Mokrosz, M.J., Bojarski, A.J., Duszyńska, B., Tatarczyńska, E., Kłodzińska, A., Dereń-Wesołek, A., Charakchieva-Minol, S., Chojnacka-Wójcik, E.
DOI: 10.1016/S0968-0896(98)00238-7
Structure-activity relationship studies of CNS agents. Part 33 - Crystal and molecular structure of 4-[omega-(benzotriazolyl)alkyl]-1-(2-methoxyphenyl)piperazines with a different pharmacological activity
Karolak-Wojciechowska, J, Fruzinski, A, Bojarski, AJ, Paluchowska, MH, Mokrosz, MJ
DOI: 10.1002/(SICI)1521-4184(199810)331:10<299::AID-ARDP299>3.3.CO;2-V
Determination of hydrophobicity of some n-alkyl derivatives of 1,2,3,4-tetrahydroisoquinoline by reversed-phase thin-layer chromatography
Kepczynska, E, Bojarski, J, Bojarski, AJ
DOI:
Determination of hydrophobicity of some N-alkyl derivatives of 1,2,3,4-tetrahydroisoquinoline by reversed-phase thin-layer chromatography
Kȩpczyńska, E., Bojarski, J., Bojarski, A.J.
DOI:
Crystal and molecular structure of 4-[ω-(benzotriazolyl)alkyl]1-(2- methoxyphenyl)piperazines with a different pharmacological activity
Karolak-Wojciechowska, J., Fruziński, A., Bojarski, A.J., Paluchowska, M.H., Mokrosz, M.J.
DOI: 10.1002/(SICI)1521-4184(199810)331:10<299::AID-ARDP299>3.0.CO;2-3
Crystal and molecular structure of N-tert-butyl-3[4-(2-methoxyphenyl)-1-piperazinyl]-2-phenylpropanamide dihydrochloride (WAY-100135)
Fruzinski, A, KarolakWojciechowska, J, Mokrosz, MJ, Bojarski, AJ
DOI:
Crystal and molecular structure of N-tert-butyl-3[4-(2-methoxyphenyl)-1-piperazinyl]-2-phenylpropanamide dihydrochloride (WAY-100135)
Fruziński, A., Karolak-Wojciechowska, J., Mokrosz, M.J., Bojarski, A.J.
DOI: