Department of Medicinal Chemistry
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Department of Medicinal Chemistry

Scientific profile
- Employees
Pracownicy zakładu
Ryszard Bugno, dr
Rafał Kurczab, dr hab.
Sabina Podlewska, dr hab.
Grzegorz Satała, dr
Katarzyna Szczepańska, dr
Adam Hogendorf, dr
Katarzyna Kaczorowska, dr
Janusz Malarz, dr
Wojciech Pietruś, dr
Dawid Warszycki, dr
Aneta Kozioł
Krystyna Nędza
Achievements
- Publications
- Grants
Grant
Development of protocol for in silico design of compounds inhibit Ebola virus infection
Dawid Warszycki, PhD
Synthesis, <sup>15</sup>N NMR spectra and GIAO calculated data of the seven positional isomers of <sup>15</sup>N-labeled N,N-dimethylsulfamoylquinoline
Marciniec, K., Maślankiewicz, A., Maślankiewicz, M.J., Kurczab, R.
DOI: 10.1016/j.molstruc.2012.01.049
The multiobjective based design, synthesis and evaluation of the arylsulfonamide/amide derivatives of aryloxyethyl and arylthioethyl-piperidines and pyrrolidines as a novel class of potent 5-HT<inf>7</inf> receptor antagonists
Zajdel, P., Kurczab, R., Grychowska, K., Satała, G., Pawłowski, M., Bojarski, A.J.
DOI: 10.1016/j.ejmech.2012.07.043
Indole-like heterocyclic compounds as a new core structure in search of potential allosteric modulators of group III metabotropic glutamate receptors
Trela, Marcin, Branski, Piotr, Bojarski, Andrzej J.
DOI:
Potential antidepressant, but not antipsychotic, activity of new 2,3-dichlorophenylpiperazines containing quinoline-or isoquinoline-sulfonamide moieties in behavioral models in mice
Wrobel, D., Jastrzebska-Wiesek, M., Partyka, A., Zajdel, P., Pawlowski, M., Marciniec, K., Maslankiewicz, A., Bojarski, A. J., Satala, G., Wesolowska, A.
DOI:
Design and synthesis of novel metabotropic glutamate receptor allosteric modulators
Stankiewicz, Anna, Bugno, Ryszard, Branski, Piotr, Bojarski, Andrzej J.
DOI: 10.1016/S1734-1140(12)70804-6
The searching of novel PAM of mGluR III by Virtual Screening of commercial chemical databases
Kurczab, Rafal, Bojarski, Andrzej J.
DOI: 10.1016/S1734-1140(12)70803-4
Quinoline- and isoquinoline-sulfonamide derivatives of LCAP as potent CNS multi-receptor - 5-HT<inf>1A</inf>/5-HT<inf>2A</inf>/5-HT<inf>7</inf>and D<inf>2</inf>/D<inf>3</inf>/D<inf>4</inf>- Agents: The synthesis and pharmacological evaluation
Zajdel, P., Marciniec, K., Maślankiewicz, A., Satała, G., Duszyńska, B., Bojarski, A.J., Partyka, A., Jastrzbska-Wisek, M., Wróbel, D., Wesołowska, A., Pawłowski, M.
DOI: 10.1016/j.bmc.2011.12.039
Synthesis, anticonvulsant activity and 5-HT<inf>1A</inf>/5-HT<inf>7</inf>receptors affinity of 1-[(4-arylpiperazin-1-yl)-propyl]-succinimides
Obniska, J., Chlebek, I., Kamiński, K., Bojarski, A.J., Satała, G.
DOI: 10.1016/S1734-1140(12)70772-7
Molecular mechanism of serotonin transporter inhibition elucidated by a new flexible docking protocol
Gabrielsen, M., Kurczab, R., Ravna, A.W., Kufareva, I., Abagyan, R., Chilmonczyk, Z., Bojarski, A.J., Sylte, I.
DOI: 10.1016/j.ejmech.2011.09.056
The multiobjective based design, synthesis and evaluation of the arylsulfonamide/amide derivatives of aryloxyethyl and arylthioethyl-piperidines and pyrrolidines as a novel class of potent 5-HT<inf>7</inf>receptor antagonists
Zajdel, P., Kurczab, R., Grychowska, K., Satała, G., Pawłowski, M., Bojarski, A.J.
DOI: 10.1016/j.ejmech.2012.07.043