Achievements

  • Publications
  • Grants

Grant

Development of protocol for in silico design of compounds inhibit Ebola virus infection

Dawid Warszycki, PhD

Sulfonamides with the N-alkyl-N′-dialkylguanidine moiety as 5-HT<inf>7</inf>receptor ligands

Zajdel, P., Subra, G., Verdie, P., Gabzdyl, E., Bojarski, A.J., Duszyńska, B., Martinez, J., Pawłowski, M.

DOI: 10.1016/j.bmcl.2009.06.038

The influence of an ethylene spacer on the 5-HT<inf>1A</inf>and 5-HT<inf>2A</inf>receptor affinity of arylpiperazine derivatives of amides with N-acylated amino acids and 3-differently substituted pyrrolidine-2,5-diones

Zajdel, P., Subra, G., Verdie, P., Bojarski, A.J., Duszyńska, B., Basista, K., Obniska, J., Martinez, J., Pawłowski, M.

DOI: 10.1016/j.ejmech.2008.05.021

Synthesis and serotonin receptor activity of the arylpiperazine alkyl/propoxy derivatives of new azatricycloundecanes

Bojarski, A.J., Kuran, B., Kossakowski, J., Kozioł, A., Jagiełło-Wójtowicz, E., Chodkowska, A.

DOI: 10.1016/j.ejmech.2008.03.019

Synthesis of 4-substituted 2-(4-methylpiperazino)pyrimidines and quinazoline analogs as serotonin 5-HT<inf>2A</inf>receptor ligands

Saczewski, J., Paluchowska, A., Klenc, J., Raux, E., Barnes, S., Sullivan, S., Duszynska, B., Bojarski, A.J., Strekowskia, L.

DOI: 10.1002/jhet.236

Atomic diversity, molecular diversity, and chemical diversity: The concept of chemodiversity

Testa, B., Vistoli, G., Pedretti, A., Bojarski, A.J.

DOI: 10.1002/cbdv.200900071

The synthesis of cyclic and acyclic long-chain arylpiperazine derivatives of salicylamide as serotonin receptor ligands

Kowalski, P., Jaśkowska, J., Bojarski, A.J., Duszyńska, B.

DOI: 10.1002/jhet.5570450125

Synthesis of new arylpiperazinylalkylthiobenzimidazole, benzothiazole, or benzoxazole derivatives as potent and selective 5-HT<inf>1A</inf> serotonin receptor ligands

Siracusa, M.A., Salerno, L., Modica, M.N., Pittalà, V., Romeo, G., Amato, M.E., Nowak, M., Bojarski, A.J., Mereghetti, I., Cagnotto, A., Mennini, T.

DOI: 10.1021/jm800176x

Novel class of arylpiperazines containing N-acylated amino acids: Their synthesis, 5-HT<inf>1A</inf>, 5-HT<inf>2A</inf>receptor affinity, and in vivo pharmacological evaluation

Zajdel, P., Subra, G., Bojarski, A.J., Duszyńska, B., Tatarczyńska, E., Nikiforuk, A., Chojnacka-Wójcik, E., Pawłowski, M., Martinez, J.

DOI: 10.1016/j.bmc.2007.02.018

Fujita-Ban QSAR analysis and CoMFA study of quinoline antagonists of immunostimulatory CpG-oligodeoxynucleotides

Paliakov, E., Henary, M., Say, M., Patterson, S.E., Parker, A., Manzel, L., Macfarlane, D.E., Bojarski, A.J., Strekowski, L.

DOI: 10.1016/j.bmc.2006.09.059

See also