Professor Andrzej Bojarski, dr hab.

Professor Andrzej Bojarski, dr hab.
Achievements
- Publications
Structure‐Activity Relationship Studies of CNS Agents, XIX: Quantitative Analysis of the Alkyl Chain Effects on the 5‐HT<inf>1A</inf> and 5‐HT<inf>2</inf> Receptor Affinities of 4‐Alkyl‐1‐arylpiperazines and Their Analogs
Autorzy: Mokrosz, J.L., Mokrosz, M.J., Charakchieva‐Minol, S., Paluchowska, M.H., Bojarski, A.J., Duszyńska, B.
DOI: 10.1002/ardp.19953280210
Date: 1995-01-01
Structure‐Activity Relationship Studies of CNS Agents, Part 25: 4,6‐Di(heteroaryl)‐2‐(N‐methylpiperazino)pyrimidines as New, Potent 5‐HT<inf>2A</inf> Receptor Ligands: A Verification of the Topographic Model
Autorzy: Mokrosz, M.J., Strekowski, L., Kozak, W.X., Duszyńska, B., Bojarski, A.J., Kłodzinska, A., Czarny, A., Cegła, M.T., Dereń‐Wesołek, A., Chojnacka‐Wójcik, E., Dove, S., Mokrosz, J.L.
DOI: 10.1002/ardp.19953280906
Date: 1995-01-01
Structure and spectral properties of β-carbolines. 8. Mechanism of the Pictet-Spengler cyclization: An MNDO approach
Autorzy: Kowalski, P., Bojarski, A.J., Mokrosz, J.L.
DOI: 10.1016/0040-4020(95)00022-Z
Date: 1995-01-01
STRUCTURE AND SPECTRAL PROPERTIES OF BETA-CARBOLINES .7. THE PICTET-SPENGLER REACTION OF TRYPTAMINES WITH N-BENZYL-4-PIPERIDONE
Autorzy: MOKROSZ, MJ, KOWALSKI, P, BOJARSKI, AJ, MOKROSZ, JL
DOI:
Date: 1994-01-01
STRUCTURE-ACTIVITY RELATIONSHIP STUDIES OF CNS AGENTS .10. 1-ARYL-2-[3-(4-ARYL-1-PIPERAZINYL)PROPYL]-1,4-DIHYDRO-3(2H)-ISOQUINOLINONES - 2 MODES OF THE INTERACTION WITH THE 5-HT(1A) RECEPTOR-SITE
Autorzy: MOKROSZ, JL, BOJARSKI, AJ, MACKOWIAK, M, BIELECKA, Z, BOKSA, J
DOI:
Date: 1994-01-01
STRUCTURE-ACTIVITY RELATIONSHIP STUDIES OF CNS AGENTS .14. STRUCTURAL REQUIREMENTS FOR THE 5-HT1A AND 5-HT2A RECEPTOR SELECTIVITY OF SIMPLE 1-(2-PYRIMIDINYL)PIPERAZINE DERIVATIVES
Autorzy: MOKROSZ, JL, STREKOWSKI, L, DUSZYNSKA, B, HARDEN, DB, MOKROSZ, MJ, BOJARSKI, AJ
DOI:
Date: 1994-01-01
STRUCTURE-ACTIVITY RELATIONSHIP STUDIES OF CNS AGENTS .16. A LOWER LIMIT OF A DISTANCE BETWEEN CRUCIAL PHARMACOPHORES OF 5-HT1A LIGANDS
Autorzy: MOKROSZ, JL, MOKROSZ, MJ, BOJARSKI, AJ, CHARAKCHIEVAMINOL, S
DOI:
Date: 1994-01-01
Structure and spectral properties of β-carbolines. Part 7. The Pictet-Spengler reaction of tryptamines with N-benzyl-4-piperidone
Autorzy: Mokrosz, M.J., Kowalski, P., Bojarski, A.J., Mokrosz, J.L.
DOI:
Date: 1994-01-01
Structure-activity relationship studies of CNS agents. Part 14: Structural requirements for the 5-HT(1A) and 5-HT(2A) receptor selectivity of simple 1-(2-pyrimidinyl)piperazine derivatives
Autorzy: Mokrosz, J.L., Strekowski, L., Duszynska, B., Harden, D.B., Mokrosz, M.J., Bojarski, A.J.
DOI:
Date: 1994-01-01
Structure-activity relationship studies OF CNS agents. Part 10: 1-Aryl-2-[3-(4-aryl-1-piperazinyl)propyl]-1,4-dihydro-3(2H)-isoquinoli nones: Two modes of the interaction with the 5-HT(1A) receptor site
Autorzy: Mokrosz, J.L., Bojarski, A.J., Mackowiak, M., Bielecka, Z., Boksa, J.
DOI:
Date: 1994-01-01