Professor Andrzej Bojarski, dr hab.

Professor Andrzej Bojarski, dr hab.

+48 12 6623365
room 325

Achievements

  • Publications

Sonication-Assisted Synthesis of (E)-2-Methyl-but-2-enyl Nucleoside Phosphonate Prodrugs

Autorzy: Bessières, M., Sari, O., Roy, V., Warszycki, D., Bojarski, A.J., Nolan, S.P., Snoeck, R., Andrei, G., Schinazi, R.F., Agrofoglio, L.A.

DOI: 10.1002/slct.201600879
Date: 2016-01-01

Erratum: Synthesis of Some Aminophosphonates Bearing N-(Fluorophenyl)-piperazynyl Moiety and Their Activity toward Serotonin Receptors (Heteroatom Chemistry (2015) 26:4 (290-298) DOI: 10.1002/hc.21259)

Autorzy: Lewki, J., Jóźwiak, A., Tokarz, P., Zagórski, P.M., Cal, D., Satała, G., Bojarski, A.J.

DOI: 10.1002/hc.21312
Date: 2016-01-01

Halogen bonding enhances activity in a series of dual 5-HT<inf>6</inf>/D<inf>2</inf>ligands designed in a hybrid bioisostere generation/virtual screening protocol

Autorzy: Staroń, J., Warszycki, D., Kurczab, R., Satała, G., Bugno, R., Hogendorf, A., Bojarski, A.J.

DOI: 10.1039/c6ra08714k
Date: 2016-01-01

GPCRdb: the G protein-coupled receptor database – an introduction

Autorzy: Munk, C., Isberg, V., Mordalski, S., Harpsøe, K., Rataj, K., Hauser, A.S., Kolb, P., Bojarski, A.J., Vriend, G., Gloriam, D.E.

DOI: 10.1111/bph.13509
Date: 2016-01-01

Concentration-Dependent Dual Mode of Zn Action at Serotonin 5-HT1A Receptors: In Vitro and In Vivo Studies

Autorzy: Satała, G., Duszyńska, B., Stachowicz, K., Rafalo, A., Pochwat, B., Luckhart, C., Albert, P.R., Daigle, M., Tanaka, K.F., Hen, R., Lenda, T., Nowak, G., Bojarski, A.J., Szewczyk, B.

DOI: 10.1007/s12035-015-9586-3
Date: 2016-01-01

Towards new 5-HT<inf>7</inf>antagonists among arylsulfonamide derivatives of (aryloxy)ethyl-alkyl amines: Multiobjective based design, synthesis, and antidepressant and anxiolytic properties

Autorzy: Canale, V., Kurczab, R., Partyka, A., Sataa, G., Ledna, T., Jastrzebska-Wiesek, M., Wesoowska, A., Bojarski, A.J., Zajdel, P.

DOI: 10.1016/j.ejmech.2015.11.040
Date: 2016-01-01

N1-Azinylsulfonyl-1H-indoles: 5-HT6 Receptor Antagonists with Procognitive and Antidepressant-Like Properties

Autorzy: Zajdel, P., Marciniec, K., Satała, G., Canale, V., Kos, T., Partyka, A., Jastrzȩbska-Wiȩsek, M., Wesołowska, A., Basińska-Ziobroń, A., Wójcikowski, J., Daniel, W.A., Bojarski, A.J., Popik, P.

DOI: 10.1021/acsmedchemlett.6b00056
Date: 2016-01-01

N-Alkylated arylsulfonamides of (aryloxy)ethyl piperidines: 5-HT<inf>7</inf>receptor selectivity versus multireceptor profile

Autorzy: Canale, V., Kurczab, R., Partyka, A., Satała, G., Słoczyńska, K., Kos, T., Jastrzębska-Więsek, M., Siwek, A., Pękala, E., Bojarski, A.J., Wesołowska, A., Popik, P., Zajdel, P.

DOI: 10.1016/j.bmc.2015.11.041
Date: 2016-01-01

Synthesis and structure-activity relationship analysis of 5-HT<inf>7</inf> receptor antagonists: Piperazin-1-yl substituted unfused heterobiaryls

Autorzy: Strekowski, L., Saczewski, J., Raux, E.A., Fernando, N.T., Klenc, J., Paranjpe, S., Raszkiewicz, A., Blake, A.L., Ehalt, A.J., Barnes, S., Baranowski, T.C., Sullivan, S.M., Satała, G., Bojarski, A.J.

DOI: 10.3390/molecules21040433
Date: 2016-01-01

Novel 1H-Pyrrolo[3,2-c]quinoline Based 5-HT<inf>6</inf>Receptor Antagonists with Potential Application for the Treatment of Cognitive Disorders Associated with Alzheimer's Disease

Autorzy: Grychowska, K., Satała, G., Kos, T., Partyka, A., Colacino, E., Chaumont-Dubel, S., Bantreil, X., Wesołowska, A., Pawłowski, M., Martinez, J., Marin, P., Subra, G., Bojarski, A.J., Lamaty, F., Popik, P., Zajdel, P.

DOI: 10.1021/acschemneuro.6b00090
Date: 2016-01-01

See also