Professor Andrzej Bojarski, dr hab.

Professor Andrzej Bojarski, dr hab.
Achievements
- Publications
PRELIMINARY EVALUATION OF CENTRAL NERVOUS SYSTEM ACTIVITY OF (<i>E</i>)-<i>N</i>-2-METHYL-3-PHENYLPROP-2-ENYL ((<i>E</i>)-<i>N</i>-α-METHYLCIN-NAMYL) DERIVATIVES OF SELECTED AMINOALKANOLS
Autorzy: Gunia-Krzyzak, Agnieszka, Pytka, Karolina, Sloczynska, Karolina, Waszkielewicz, Anna. M., Satala, Grzegorz, Bojarski, Andrzej J., Sapa, Jacek, Filipek, Barbara, Cegla, Marek, Pekala, Elzbieta, Marona, Henryk
DOI:
Date: 2016-01-01
IP562083 a novel mGluR7 negative allosteric modulator
Autorzy: Branski, Piotr, Burnat, Grzegorz, Stankiewicz, Anna, Bugno, Ryszard, Paluchowska, Maria, Kaczorowska, Katarzyna, Chruscicka, Barbara, Bojarski, Andrzej, Pilc, Andrzej
DOI: 10.1016/J.PHAREP.2015.06.055
Date: 2015-01-01
Ligand-Based Virtual Screening in a Search for Novel Anti-HIV-1 Chemotypes
Autorzy: Kurczyk, A., Warszycki, D., Musiol, R., Kafel, R., Bojarski, A.J., Polanski, J.
DOI: 10.1021/acs.jcim.5b00295
Date: 2015-01-01
Antidepressant- and anxiolytic-like activity of 7-phenylpiperazinylalkyl-1,3-dimethyl-purine-2,6-dione derivatives with diversified 5-HT<inf>1A</inf>receptor functional profile
Autorzy: Partyka, A., Chłoń-Rzepa, G., Wasik, A., Jastrzębska-Więsek, M., Bucki, A., Kołaczkowski, M., Satała, G., Bojarski, A.J., Wesołowska, A.
DOI: 10.1016/j.bmc.2014.11.008
Date: 2015-01-01
Novel 4-aryl-pyrido[1,2-c]pyrimidines with dual SSRI and 5-HT<inf>1A</inf> activity. part 5
Autorzy: Gomolka, A., Ciesielska, A., Wróbel, M.Z., Chodkowski, A., Kleps, J., Dawidowski, M., Siwek, A., Wolak, M., Stachowicz, K., Slawinska, A., Nowak, G., Satala, G., Bojarski, A.J., Belka, M., Ulenberg, S., Baczek, T., Skowronek, P., Turlo, J., Herold, F.
DOI: 10.1016/j.ejmech.2015.05.003
Date: 2015-01-01
Arylsulfonamide derivatives of (aryloxy)ethylpiperidines as selective 5-HT<inf>7</inf>receptor antagonists and their psychotropic properties
Autorzy: Zajdel, P., Canale, V., Partyka, A., Marciniec, K., Kurczab, R., Satała, G., Siwek, A., Jastrzębska-Więsek, M., Wesołowska, A., Kos, T., Popik, P., Bojarski, A.J.
DOI: 10.1039/c5md00166h
Date: 2015-01-01
Towards novel 5-HT<inf>7</inf>versus 5-HT<inf>1A</inf>receptor ligands among LCAPs with cyclic amino acid amide fragments: Design, synthesis, and antidepressant properties. Part II
Autorzy: Canale, V., Kurczab, R., Partyka, A., SataÅa, G., Witek, J., Jastrzäbska-Wiäsek, M., Pawåowski, M., Bojarski, A.J., WesoÅowska, A., Zajdel, P.
DOI: 10.1016/j.ejmech.2014.12.041
Date: 2015-01-01
Solid-Supported Synthesis and 5-HT<inf>7</inf>/5-HT<inf>1A</inf> Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1H)-one
Autorzy: Grychowska, K., Masurier, N., Verdié, P., Satała, G., Bojarski, A.J., Martinez, J., Pawłowski, M., Subra, G., Zajdel, P.
DOI: 10.1111/cbdd.12539
Date: 2015-01-01
Structure-5-HT Receptor Affinity Relationship in a New Group of 7-Arylpiperazynylalkyl and 7-Tetrahydroisoquinolinylalkyl Derivatives of 8-Amino-1,3-dimethyl-1H-purine-2,6(3H,7H)-dione
Autorzy: Zmudzki, P., Chłoń-Rzepa, G., Bojarski, A.J., Zygmunt, M., Kazek, G., Mordyl, B., Pawłowski, M.
DOI: 10.1002/ardp.201400392
Date: 2015-01-01
Structure-activity relationships and molecular studies of novel arylpiperazinylalkyl purine-2,4-diones and purine-2,4,8-triones with antidepressant and anxiolytic-like activity
Autorzy: Zagórska, A., Kolaczkowski, M., Bucki, A., Siwek, A., Kazek, G., Satala, G., Bojarski, A.J., Partyka, A., Wesolowska, A., Pawlowski, M.
DOI: 10.1016/j.ejmech.2015.04.046
Date: 2015-01-01