Professor Andrzej Bojarski, dr hab.

Professor Andrzej Bojarski, dr hab.

+48 12 6623365
room 325

Achievements

  • Publications

RECEPTOR AFFINITY AND PHOSPHODIESTERASES 4B AND 10A ACTIVITY OF OCTAHYDRO- AND 6,7-DIMETHOXY-3,4-DIHYDRO-ISOQUINOLIN-2(1H)-YL-ALKYL DERIVATIVES OF IMIDAZO- AND PYRIMIDINO[2,1-f]PURINES

Autorzy: Zagorska, Agnieszka, Gryzlo, Beata, Satala, Grzegorz, Bojarski, Andrzej J., Gluch-Lutwin, Monika, Mordyl, Barbara, Kazek, Grzegorz, Pawlowski, Maciej

DOI:
Date: 2016-01-01

NEW SPIROHYDANTOIN DERIVATIVES - SYNTHESIS, PHARMACOLOGICAL EVALUATION, AND MOLECULAR MODELING STUDY

Autorzy: Czopek, Anna, Zagorska, Agnieszka, Kolaczkowski, Marcin, Bucki, Adam, Gryzlo, Beata, Rychtyk, Joanna, Pawlowski, Maciej, Siwek, Agata, Satala, Grzegorz, Bojarskp, Andrzej, Kubacka, Monika, Filipek, Barbara

DOI:
Date: 2016-01-01

Preliminary evaluation of central nervous system activity of (E)-N-2-methyl-3-phenylprop-2-enyl ((E)-N- α-methylcinnamyl) derivatives of selected aminoalkanols

Autorzy: Gunia-Krzyzak, A., Pytka, K., Słoczyńska, K., Waszkielewicz, A.M., Satała, G., Bojarski, A.J., Sapa, J., Filipek, B., Cegła, M., Pekala, E., Marona, H.

DOI:
Date: 2016-01-01

Receptor affinity and phosphodiesterases 4B and 10A activity of octahydro- and 6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl-alkyl derivatives of imidazo- and pyrimidino[2,1-f]purines

Autorzy: Zagórska, A., Gryzło, B., Satała, G., Bojarski, A.J., Głuch-Lutwin, M., Mordyl, B., Kazek, G., Pawłowski, M.

DOI:
Date: 2016-01-01

New spirohydantoin derivatives - Synthesis, pharmacological evaluation, and molecular modeling study

Autorzy: Czopek, A., Zagórska, A., Kołaczkowski, M., Bucki, A., Gryzło, B., Rychtyk, J., Pawłowski, M., Siwek, A., Satała, G., Bojarski, A., Kubacka, M., Filipek, B.

DOI:
Date: 2016-01-01

Structural modifications of the serotonin 5-HT<inf>7</inf>receptor agonist N -(4-cyanophenylmethyl)-4-(2-biphenyl)-1-piperazinehexanamide (LP-211) to improve in vitro microsomal stability: A case study

Autorzy: Lacivita, E., Podlewska, S., Speranza, L., Niso, M., Satała, G., Perrone, R., Perrone-Capano, C., Bojarski, A.J., Leopoldo, M.

DOI: 10.1016/j.ejmech.2016.05.005
Date: 2016-01-01

Straightforward synthesis of 2,4,6-trisubstituted 1,3,5-triazine compounds targeting cysteine cathepsins K and S

Autorzy: Plebanek, E., Chevrier, F., Roy, V., Garenne, T., Lecaille, F., Warszycki, D., Bojarski, A.J., Lalmanach, G., Agrofoglio, L.A.

DOI: 10.1016/j.ejmech.2016.05.009
Date: 2016-01-01

Rational design in search for 5-phenylhydantoin selective 5-HT<inf>7</inf>R antagonists. Molecular modeling, synthesis and biological evaluation

Autorzy: Kucwaj-Brysz, K., Warszycki, D., Podlewska, S., Witek, J., Witek, K., Izquierdo, A.G., Satała, G., Loza, M.I., Lubelska, A., Latacz, G., Bojarski, A.J., Castro, M., Kieć-Kononowicz, K., Handzlik, J.

DOI: 10.1016/j.ejmech.2016.02.024
Date: 2016-01-01

Structure–5-HT/D<inf>2</inf>Receptor Affinity Relationship in a New Group of 1-Arylpiperazynylalkyl Derivatives of 8-Dialkylamino-3,7-dimethyl-1H-purine-2,6(3H,7H)-dione

Autorzy: Żmudzki, P., Satała, G., Chłoń-Rzepa, G., Bojarski, A.J., Kazek, G., Siwek, A., Gryboś, A., Głuch-Lutwin, M., Wesołowska, A., Pawłowski, M.

DOI: 10.1002/ardp.201600162
Date: 2016-01-01

GPCRdb: An information system for G protein-coupled receptors

Autorzy: Isberg, V., Mordalski, S., Munk, C., Rataj, K., Harpsøe, K., Hauser, A.S., Vroling, B., Bojarski, A.J., Vriend, G., Gloriam, D.E.

DOI: 10.1093/nar/gkv1178
Date: 2016-01-01

See also