Publications

Scientific activity

Synthesis, antidepressant evaluation and docking studies of long-chain alkylnitroquipazines as serotonin transporter inhibitors

Autorzy: Gabrielsen, M., Wolosewicz, K., Zawadzka, A., Kossakowski, J., Nowak, G., Wolak, M., Stachowicz, K., Siwek, A., Ravna, A.W., Kufareva, I., Kozerski, L., Bednarek, E., Sitkowski, J., Bocian, W., Abagyan, R., Bojarski, A.J., Sylte, I., Chilmonczyk, Z.

DOI: 10.1111/cbdd.12116
Date: 2013-01-01

Novel mannich bases, 5-arylimidazolidine-2,4-dione derivatives with dual 5-HT<inf>1A</inf> receptor and serotonin transporter affinity

Autorzy: Czopek, A., Kołaczkowski, M., Bucki, A., Byrtus, H., Pawłowski, M., Siwek, A., Bojarski, A.J., Bednarski, M., Wróbel, D., Wesołowska, A.

DOI: 10.1002/ardp.201200378
Date: 2013-01-01

Synthesis and biological evaluation of novel pyrrolidine-2,5-dione derivatives as potential antidepressant agents. Part 1

Autorzy: Wróbel, M.Z., Chodkowski, A., Herold, F., Gomółka, A., Kleps, J., Mazurek, A.P., Pluciński, F., Mazurek, A., Nowak, G., Siwek, A., Stachowicz, K., Sławińska, A., Wolak, M., Szewczyk, B., Satała, G., Bojarski, A.J., Turło, J.

DOI: 10.1016/j.ejmech.2013.02.033
Date: 2013-01-01

A multidimensional analysis of machine learning methods performance in the classification of bioactive compounds

Autorzy: Smusz, S., Kurczab, R., Bojarski, A.J.

DOI: 10.1016/j.chemolab.2013.08.003
Date: 2013-01-01

Quinolinesulfonamides of aryloxy-/arylthio-ethyl piperidines: Influence of an arylether fragment on 5-HT<inf>1A</inf>/5-HT<inf>7</inf> receptor selectivity

Autorzy: Grychowska, K., Marciniec, K., Canale, V., Szymiec, M., Glanowski, G., Satała, G., Maślankiewicz, A., Pawłowski, M., Bojarski, A.J., Zajdel, P.

DOI: 10.1002/ardp.201200322
Date: 2013-01-01

New strategy for receptor-based pharmacophore query construction: A case study for 5-HT<inf>7</inf> receptor ligands

Autorzy: Kurczab, R., Bojarski, A.J.

DOI: 10.1021/ci4005207
Date: 2013-01-01

New 8-aminoalkyl derivatives of purine-2,6-dione with arylalkyl, allyl or propynyl substituents in position 7, their 5-HT<inf>1A</inf>, 5-HT<inf>2A</inf>, and 5-HT<inf>7</inf>receptor affinity and pharmacological evaluation

Autorzy: Chłoń-Rzepa, G., Zmudzki, P., Satała, G., Duszyńska, B., Partyka, A., Wróbel, D., Jastrzȩbska-Wiȩsek, M., Wesołowska, A., Bojarski, A.J., Pawłowski, M., Zajdel, P.

DOI: 10.1016/S1734-1140(13)70960-5
Date: 2013-01-01

Synthesis and evaluation of pharmacological properties of some new xanthone derivatives with piperazine moiety

Autorzy: Waszkielewicz, A.M., Gunia, A., Szkaradek, N., Pytka, K., Siwek, A., Satała, G., Bojarski, A.J., Szneler, E., Marona, H.

DOI: 10.1016/j.bmcl.2013.05.062
Date: 2013-01-01

A linear combination of pharmacophore hypotheses as a new tool in search of new active compounds - An application for 5-HT<inf>1A</inf>receptor ligands

Autorzy: Warszycki, D., Mordalski, S., Kristiansen, K., Kafel, R., Sylte, I., Chilmonczyk, Z., Bojarski, A.J.

DOI: 10.1371/journal.pone.0084510
Date: 2013-01-01

Morphine-induced place preference affects mRNA expression of G protein α subunits in rat brain

Autorzy: Zelek-Molik, A., Bielawski, A., Kreiner, G., Popik, P., Vetulani, J., Nalepa, I.

DOI: 10.1016/S1734-1140(12)70850-2
Date: 2012-01-01

See also