dr Dawid Warszycki

dr Dawid Warszycki

+48 12 6623301
pokój 326
Zakład Chemii Leków

Dokonania naukowe

  • Publikacje

Novel Tripeptides as Tyrosinase Inhibitors: In Silico and In Vitro Approaches

Autorzy: Michał Dymek, Dawid Warszycki, Sabina Podlewska, Elżbieta Sikora

DOI: 10.3390/ijms252413509
Date: 2024-12-17

Isomeric Activity Cliffs—A Case Study for Fluorine Substitution of Aminergic G Protein-Coupled Receptor Ligands

Autorzy: Wojciech Pietruś, Rafał Kurczab, Dawid Warszycki, Andrzej J. Bojarski, Jürgen Bajorath

DOI: 10.3390/molecules28020490
Date: 2023-01-04

Improved HDAC Inhibition, Stronger Cytotoxic Effect and Higher Selectivity against Leukemias and Lymphomas of Novel, Tricyclic Vorinostat Analogues

Autorzy: Bartosz Bieszczad, Damian Garbicz, Marta Świtalska, Marta K. Dudek, Dawid Warszycki, Joanna Wietrzyk, Elżbieta Grzesiuk, Adam Mieczkowski

DOI: 10.3390/ph14090851
Date: 2021-08-26

Novel Vorinostat Analogues with Improved HDAC Inhibition, Stronger Cytotoxic Effect and Higher Selectivity Against Leukemias and Lymphomas

Autorzy: Bartosz Bieszczad, Damian Garbicz, Marta Świtalska, Marta K. Dudek, Dawid Warszycki, Joanna Wietrzyk, Elżbieta Grzesiuk, Adam Mieczkowski

DOI: 10.20944/preprints202105.0251.v1
Date: 2021-05-11

Design, synthesis and biological evaluation of 2-substituted-6-[(4-substituted-1-piperidyl)methyl]-1H-benzimidazoles as inhibitors of ebola virus infection

Autorzy: Maxime Bessières, Elżbieta Plebanek, Payel Chatterjee, Punya Shrivastava-Ranjan, Mike Flint, Christina F. Spiropoulou, Dawid Warszycki, Andrzej J. Bojarski, Vincent Roy, Luigi A. Agrofoglio

DOI: 10.1016/j.ejmech.2021.113211
Date: 2021-03-01

Rationally designed N-phenylsulfonylindoles as a tool for the analysis of the non-basic 5-HT<sub>6</sub>R ligands binding mode.

Autorzy:

DOI: 10.1016/j.ejmech.2020.112916
Date: 2020-10-09

Virtual screening-driven discovery of dual 5-HT<sub>6</sub>/5-HT<sub>2A</sub> receptor ligands with pro-cognitive properties.

Autorzy:

DOI: 10.1016/j.ejmech.2019.111857
Date: 2019-11-07

In Silico Methods for the Discovery of Orthosteric GABA<sub>B</sub> Receptor Compounds

Autorzy: Linn M. Evenseth, Dawid Warszycki, Andrzej Bojarski, Mari Gabrielsen, Ingebrigt Sylte

DOI: 10.3390/molecules24050935
Date: 2019-03-01

The effect of the intramolecular C-H⋯O interactions on the conformational preferences of bis-arylsulfones-5-HT<inf>6</inf>receptor antagonists and beyond

Autorzy: Kalinowska-Tłuścik, J., Staroń, J., Krawczuk, A., Mordalski, S., Warszycki, D., Satała, G., Hogendorf, A.S., Bojarski, A.J.

DOI: 10.1039/c8ra03107j
Date: 2018-01-01

Selective inhibition of human cathepsin S by 2,4,6-trisubstituted 1,3,5-triazine analogs

Autorzy: Tber, Z., Wartenberg, M., Jacques, J.-E., Roy, V., Lecaille, F., Warszycki, D., Bojarski, A.J., Lalmanach, G., Agrofoglio, L.A.

DOI: 10.1016/j.bmc.2018.07.032
Date: 2018-01-01

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